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Found 16 Enz. Inhib. hit(s) with all data for entry = 50041821
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50416331(CHEMBL1170167)
Affinity DataKi:  1.74nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO-A1 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50416330(CHEMBL1170166)
Affinity DataKi:  2.34nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50416331(CHEMBL1170167)
Affinity DataKi:  3.55nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50416325(CHEMBL1170990)
Affinity DataKi:  21.9nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50416334(CHEMBL1171380)
Affinity DataKi:  30.9nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50416332(CHEMBL1172502)
Affinity DataKi:  31.6nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50416333(CHEMBL1171379)
Affinity DataKi:  40.7nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50416330(CHEMBL1170166)
Affinity DataKi:  75.9nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO-A1 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50416329(CHEMBL1169972)
Affinity DataKi:  79.4nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50416335(CHEMBL1170168)
Affinity DataKi:  97.7nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50416326(CHEMBL1169969)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50416328(CHEMBL1169971)
Affinity DataKi:  115nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50416333(CHEMBL1171379)
Affinity DataKi:  182nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO-A1 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50416333(CHEMBL1171379)
Affinity DataKi:  708nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in human HeLa cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50416327(CHEMBL1169970)
Affinity DataKi:  1.05E+3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade De A Coru£A

Curated by ChEMBL
LigandPNGBDBM50416330(CHEMBL1170166)
Affinity DataKi:  6.46E+3nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in human HeLa cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed