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Found 9 Enz. Inhib. hit(s) with all data for entry = 50041804
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50415880(CHEMBL1097489)
Affinity DataKi:  15.8nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 60 mins by beta scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50415880(CHEMBL1097489)
Affinity DataKi:  158nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in forskolin-stimulated CHO cells assessed as inhibition of NSCA-induced decrease in cAM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50415879(CHEMBL1099202)
Affinity DataKi:  316nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells after 180 mins by beta scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50415879(CHEMBL1099202)
Affinity DataKi:  501nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in forskolin-stimulated CHO cells assessed as inhibition of NSCA-induced decrease in cAM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50415878(CHEMBL1095872)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 30 mins by beta scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50415878(CHEMBL1095872)
Affinity DataKi:  2.00E+3nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in HEK293 cells assessed as inhibition of NSCA-induced cAMP accumulation pre-incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50415881(CHEMBL1097859)
Affinity DataKi:  2.51E+3nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in human HeLa cells after 30 mins by beta scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50415881(CHEMBL1097859)
Affinity DataKi:  3.16E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells after 180 mins by beta scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universidade Do Minho

Curated by ChEMBL
LigandPNGBDBM50415881(CHEMBL1097859)
Affinity DataKi:  7.94E+3nMAssay Description:Antagonist activity at human adenosine A2A receptor expressed in CHO cells assessed as inhibition of NSCA-induced cAMP accumulation pre-incubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed