Compile Data Set for Download or QSAR
maximum 50k data
Found 66 Enz. Inhib. hit(s) with all data for entry = 50031784
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319102(5-(3,5-difluorophenyl)-2-(3-(6-hydroxynaphthalen-2...)
Affinity DataIC50:  3nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50313977(2-(3-(3-(5-hydroxypyridin-2-yl)-1,2,4-oxadiazol-5-...)
Affinity DataIC50:  4nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319109(2-(3-(3-(5-hydroxypyridin-2-yl)-1,2,4-oxadiazol-5-...)
Affinity DataIC50:  4nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319123((4S,5R)-2-(3-(3-(5-fluoropyridin-2-yl)-1,2,4-oxadi...)
Affinity DataIC50:  6nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319096(5-butyl-2-(3-(6-hydroxynaphthalen-2-yl)propanamido...)
Affinity DataIC50:  6nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319110(5-(3-fluorophenyl)-2-(3-(3-(5-hydroxypyridin-2-yl)...)
Affinity DataIC50:  7nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319100(5-(3-fluorophenyl)-2-(3-(6-hydroxynaphthalen-2-yl)...)
Affinity DataIC50:  7.40nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50271314(2-(3-(6-hydroxynaphthalen-2-yl)propanamido)cyclohe...)
Affinity DataIC50:  8nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319095(2-(3-(6-hydroxynaphthalen-2-yl)propanamido)-5-prop...)
Affinity DataIC50:  8nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319113((4S,5R)-5-(3-fluorophenyl)-2-(3-(3-(5-hydroxypyrid...)
Affinity DataIC50:  8nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319101(5-(4-fluorophenyl)-2-(3-(6-hydroxynaphthalen-2-yl)...)
Affinity DataIC50:  8.60nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319120(2-(3-(3-(5-fluoropyridin-2-yl)-1,2,4-oxadiazol-5-y...)
Affinity DataIC50:  9nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319111(5-(6-fluoropyridin-3-yl)-2-(3-(3-(5-hydroxypyridin...)
Affinity DataIC50:  9nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319099(5-(2-fluorophenyl)-2-(3-(6-hydroxynaphthalen-2-yl)...)
Affinity DataIC50:  11nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319112((4S,5R)-2-(3-(3-(5-hydroxypyridin-2-yl)-1,2,4-oxad...)
Affinity DataIC50:  12nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319106(2-(3-(6-hydroxynaphthalen-2-yl)propanamido)-5-(1-m...)
Affinity DataIC50:  14nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319121(2-(2-amino-3-(3-(5-fluoropyridin-2-yl)-1,2,4-oxadi...)
Affinity DataIC50:  15nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319104(5-(6-fluoropyridin-3-yl)-2-(3-(6-hydroxynaphthalen...)
Affinity DataIC50:  16nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319105(2-(3-(6-hydroxynaphthalen-2-yl)propanamido)-5-(6-(...)
Affinity DataIC50:  18nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319118(5-(3,5-difluorophenyl)-2-(3-(3-(5-fluoropyridin-2-...)
Affinity DataIC50:  19nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319119(2-(2-amino-3-(3-(5-fluoropyridin-2-yl)-1,2,4-oxadi...)
Affinity DataIC50:  28nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319115(2-(2-amino-3-(3-(5-fluoropyridin-2-yl)-1,2,4-oxadi...)
Affinity DataIC50:  32nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319097(2-(3-(6-hydroxynaphthalen-2-yl)propanamido)-5-phen...)
Affinity DataIC50:  34nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319114(2-(3-(3-(5-fluoropyridin-2-yl)-1,2,4-oxadiazol-5-y...)
Affinity DataIC50:  35nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319108(5-(2-fluoropyridin-3-yl)-2-(3-(4'-hydroxybiphenyl-...)
Affinity DataIC50:  36nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319094(2-(3-(6-hydroxynaphthalen-2-yl)propanamido)-5-meth...)
Affinity DataIC50:  43nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319103(5-(2-fluoropyridin-3-yl)-2-(3-(6-hydroxynaphthalen...)
Affinity DataIC50:  52nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319116(5-(3-fluorophenyl)-2-(3-(3-(5-fluoropyridin-2-yl)-...)
Affinity DataIC50:  57nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319117(2-(2-amino-3-(3-(5-fluoropyridin-2-yl)-1,2,4-oxadi...)
Affinity DataIC50:  85nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319107(2-(3-(6-hydroxynaphthalen-2-yl)propanamido)-5-(1-m...)
Affinity DataIC50:  120nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM23515(CHEMBL573 | Niacin | Nicotinic Acid | [5, 6-3H]-ni...)
Affinity DataIC50:  140nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319122(2-(3-(3-(5-fluoropyridin-2-yl)-1,2,4-oxadiazol-5-y...)
Affinity DataIC50:  280nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319098(5-hydroxy-2-(3-(6-hydroxynaphthalen-2-yl)propanami...)
Affinity DataIC50:  420nMAssay Description:Displacement of [3H]niacin from human niacin receptor expressed in CHO-KI cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319114(2-(3-(3-(5-fluoropyridin-2-yl)-1,2,4-oxadiazol-5-y...)
Affinity DataEC50:  490nMAssay Description:Agonist activity at human niacin receptor expressed in CHO-KI cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319115(2-(2-amino-3-(3-(5-fluoropyridin-2-yl)-1,2,4-oxadi...)
Affinity DataEC50:  460nMAssay Description:Agonist activity at human niacin receptor expressed in CHO-KI cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319116(5-(3-fluorophenyl)-2-(3-(3-(5-fluoropyridin-2-yl)-...)
Affinity DataEC50:  230nMAssay Description:Agonist activity at human niacin receptor expressed in CHO-KI cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319117(2-(2-amino-3-(3-(5-fluoropyridin-2-yl)-1,2,4-oxadi...)
Affinity DataEC50:  250nMAssay Description:Agonist activity at human niacin receptor expressed in CHO-KI cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319118(5-(3,5-difluorophenyl)-2-(3-(3-(5-fluoropyridin-2-...)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human niacin receptor expressed in CHO-KI cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319119(2-(2-amino-3-(3-(5-fluoropyridin-2-yl)-1,2,4-oxadi...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human niacin receptor expressed in CHO-KI cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319120(2-(3-(3-(5-fluoropyridin-2-yl)-1,2,4-oxadiazol-5-y...)
Affinity DataEC50:  45nMAssay Description:Agonist activity at human niacin receptor expressed in CHO-KI cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319121(2-(2-amino-3-(3-(5-fluoropyridin-2-yl)-1,2,4-oxadi...)
Affinity DataEC50:  46nMAssay Description:Agonist activity at human niacin receptor expressed in CHO-KI cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319122(2-(3-(3-(5-fluoropyridin-2-yl)-1,2,4-oxadiazol-5-y...)
Affinity DataEC50:  7.40E+3nMAssay Description:Agonist activity at human niacin receptor expressed in CHO-KI cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319113((4S,5R)-5-(3-fluorophenyl)-2-(3-(3-(5-hydroxypyrid...)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human niacin receptor expressed in CHO-KI cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319112((4S,5R)-2-(3-(3-(5-hydroxypyridin-2-yl)-1,2,4-oxad...)
Affinity DataEC50:  6nMAssay Description:Agonist activity at human niacin receptor expressed in CHO-KI cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319111(5-(6-fluoropyridin-3-yl)-2-(3-(3-(5-hydroxypyridin...)
Affinity DataEC50:  98nMAssay Description:Agonist activity at human niacin receptor expressed in CHO-KI cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319110(5-(3-fluorophenyl)-2-(3-(3-(5-hydroxypyridin-2-yl)...)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human niacin receptor expressed in CHO-KI cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319109(2-(3-(3-(5-hydroxypyridin-2-yl)-1,2,4-oxadiazol-5-...)
Affinity DataEC50:  17nMAssay Description:Agonist activity at human niacin receptor expressed in CHO-KI cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50313977(2-(3-(3-(5-hydroxypyridin-2-yl)-1,2,4-oxadiazol-5-...)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human niacin receptor expressed in CHO-KI cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319108(5-(2-fluoropyridin-3-yl)-2-(3-(4'-hydroxybiphenyl-...)
Affinity DataEC50:  137nMAssay Description:Agonist activity at human niacin receptor expressed in CHO-KI cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50319107(2-(3-(6-hydroxynaphthalen-2-yl)propanamido)-5-(1-m...)
Affinity DataEC50:  2.65E+3nMAssay Description:Agonist activity at human niacin receptor expressed in CHO-KI cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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