Compile Data Set for Download or QSAR
maximum 50k data
Found 81 Enz. Inhib. hit(s) with all data for entry = 50031964
TargetD(1A) dopamine receptor(RAT)
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in CRL:CD(SD)BR-COBS rat striatum by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322374(1,6-bis(4-phenylpiperazin-1-yl)hexane | CHEMBL1172...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in CRL:CD(SD)BR-COBS rat striatum by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322373(1-(3-chlorophenyl)-4-(6-(4-(3-methoxyphenyl)pipera...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A receptor in rat CRL:CD(SD)BR-COBS hippocampus by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322371(1-(pyridin-2-yl)-4-(6-(4-m-tolylpiperazin-1-yl)hex...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A receptor in rat CRL:CD(SD)BR-COBS hippocampus by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322374(1,6-bis(4-phenylpiperazin-1-yl)hexane | CHEMBL1172...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A receptor in rat CRL:CD(SD)BR-COBS hippocampus by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in CRL:CD(SD)BR-COBS rat striatum by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM35254(2-methyl-4-(4-methylpiperazin-1-yl)-10H-thieno[2,3...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in CRL:CD(SD)BR-COBS rat cortex by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322373(1-(3-chlorophenyl)-4-(6-(4-(3-methoxyphenyl)pipera...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in CRL:CD(SD)BR-COBS rat striatum by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50265376(CHEMBL496739 | N-(4-(4-(m-Tolyl)piperazin-1-yl)but...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in CRL:CD(SD)BR-COBS rat striatum by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A receptor in rat CRL:CD(SD)BR-COBS hippocampus by scintillation spectrometryMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322372(1-(6-methylpyridin-2-yl)-4-(6-(4-m-tolylpiperazin-...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in CRL:CD(SD)BR-COBS rat cortex by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322373(1-(3-chlorophenyl)-4-(6-(4-(3-methoxyphenyl)pipera...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in CRL:CD(SD)BR-COBS rat cortex by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322376(1,6-bis(4-(3-methoxyphenyl)piperazin-1-yl)hexane |...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A receptor in rat CRL:CD(SD)BR-COBS hippocampus by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322380(1-(6-methylpyridin-2-yl)-4-(6-(4-phenylpiperazin-1...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A receptor in rat CRL:CD(SD)BR-COBS hippocampus by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in CRL:CD(SD)BR-COBS rat cortex by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322369(1-phenyl-4-(6-(4-m-tolylpiperazin-1-yl)hexyl)piper...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in CRL:CD(SD)BR-COBS rat cortex by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322371(1-(pyridin-2-yl)-4-(6-(4-m-tolylpiperazin-1-yl)hex...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in CRL:CD(SD)BR-COBS rat cortex by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in CRL:CD(SD)BR-COBS rat cortex by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322372(1-(6-methylpyridin-2-yl)-4-(6-(4-m-tolylpiperazin-...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A receptor in rat CRL:CD(SD)BR-COBS hippocampus by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322377(1,6-bis(4-(3-chlorophenyl)piperazin-1-yl)hexane | ...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in CRL:CD(SD)BR-COBS rat striatum by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50265376(CHEMBL496739 | N-(4-(4-(m-Tolyl)piperazin-1-yl)but...)
Affinity DataKi:  11.9nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A receptor in rat CRL:CD(SD)BR-COBS hippocampus by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50265376(CHEMBL496739 | N-(4-(4-(m-Tolyl)piperazin-1-yl)but...)
Affinity DataKi:  15.3nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in CRL:CD(SD)BR-COBS rat cortex by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322377(1,6-bis(4-(3-chlorophenyl)piperazin-1-yl)hexane | ...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A receptor in rat CRL:CD(SD)BR-COBS hippocampus by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322378(1,6-bis(4-(pyridin-2-yl)piperazin-1-yl)hexane | CH...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A receptor in rat CRL:CD(SD)BR-COBS hippocampus by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322369(1-phenyl-4-(6-(4-m-tolylpiperazin-1-yl)hexyl)piper...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A receptor in rat CRL:CD(SD)BR-COBS hippocampus by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322369(1-phenyl-4-(6-(4-m-tolylpiperazin-1-yl)hexyl)piper...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in CRL:CD(SD)BR-COBS rat striatum by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322375(1,6-bis(4-m-tolylpiperazin-1-yl)hexane | CHEMBL117...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in CRL:CD(SD)BR-COBS rat cortex by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM35254(2-methyl-4-(4-methylpiperazin-1-yl)-10H-thieno[2,3...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in CRL:CD(SD)BR-COBS rat striatum by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322380(1-(6-methylpyridin-2-yl)-4-(6-(4-phenylpiperazin-1...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in CRL:CD(SD)BR-COBS rat striatum by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322380(1-(6-methylpyridin-2-yl)-4-(6-(4-phenylpiperazin-1...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in CRL:CD(SD)BR-COBS rat cortex by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322376(1,6-bis(4-(3-methoxyphenyl)piperazin-1-yl)hexane |...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in CRL:CD(SD)BR-COBS rat striatum by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322376(1,6-bis(4-(3-methoxyphenyl)piperazin-1-yl)hexane |...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in CRL:CD(SD)BR-COBS rat cortex by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322379(1-phenyl-4-(6-(4-(pyridin-2-yl)piperazin-1-yl)hexy...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A receptor in rat CRL:CD(SD)BR-COBS hippocampus by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322374(1,6-bis(4-phenylpiperazin-1-yl)hexane | CHEMBL1172...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in CRL:CD(SD)BR-COBS rat cortex by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322372(1-(6-methylpyridin-2-yl)-4-(6-(4-m-tolylpiperazin-...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in CRL:CD(SD)BR-COBS rat striatum by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322379(1-phenyl-4-(6-(4-(pyridin-2-yl)piperazin-1-yl)hexy...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in CRL:CD(SD)BR-COBS rat striatum by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322370(4-(4-(6-(4-phenylpiperazin-1-yl)hexyl)piperazin-1-...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in CRL:CD(SD)BR-COBS rat cortex by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322379(1-phenyl-4-(6-(4-(pyridin-2-yl)piperazin-1-yl)hexy...)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in CRL:CD(SD)BR-COBS rat cortex by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM35254(2-methyl-4-(4-methylpiperazin-1-yl)-10H-thieno[2,3...)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in CRL:CD(SD)BR-COBS rat striatum by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322370(4-(4-(6-(4-phenylpiperazin-1-yl)hexyl)piperazin-1-...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in CRL:CD(SD)BR-COBS rat striatum by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322371(1-(pyridin-2-yl)-4-(6-(4-m-tolylpiperazin-1-yl)hex...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in CRL:CD(SD)BR-COBS rat striatum by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322378(1,6-bis(4-(pyridin-2-yl)piperazin-1-yl)hexane | CH...)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in CRL:CD(SD)BR-COBS rat cortex by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322375(1,6-bis(4-m-tolylpiperazin-1-yl)hexane | CHEMBL117...)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A receptor in rat CRL:CD(SD)BR-COBS hippocampus by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322370(4-(4-(6-(4-phenylpiperazin-1-yl)hexyl)piperazin-1-...)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A receptor in rat CRL:CD(SD)BR-COBS hippocampus by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322375(1,6-bis(4-m-tolylpiperazin-1-yl)hexane | CHEMBL117...)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in CRL:CD(SD)BR-COBS rat striatum by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322377(1,6-bis(4-(3-chlorophenyl)piperazin-1-yl)hexane | ...)
Affinity DataKi:  98nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in CRL:CD(SD)BR-COBS rat cortex by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50322378(1,6-bis(4-(pyridin-2-yl)piperazin-1-yl)hexane | CH...)
Affinity DataKi:  159nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in CRL:CD(SD)BR-COBS rat striatum by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A receptor in rat CRL:CD(SD)BR-COBS hippocampus by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in CRL:CD(SD)BR-COBS rat striatum by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Universita Di Siena

Curated by ChEMBL
LigandPNGBDBM50265376(CHEMBL496739 | N-(4-(4-(m-Tolyl)piperazin-1-yl)but...)
Affinity DataKi:  263nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in CRL:CD(SD)BR-COBS rat striatum by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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