Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50032035
TargetCannabinoid receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50200833(CHEMBL373626 | N-((2S,3S)-4-(4-chlorophenyl)-3-phe...)
Affinity DataIC50:  0.540nMAssay Description:Displacement of [3H]CP55490 from human recombinant cannabinoid CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323607(CHEMBL1209596 | rac-N-((2S,3S)-3-(3-bromophenyl)-4...)
Affinity DataIC50:  0.590nMAssay Description:Displacement of [3H]CP55490 from human recombinant cannabinoid CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50200841(CHEMBL220360 | MK-0364 | MK-0634 | N-((2S,3S)-4-(4...)
Affinity DataIC50:  0.740nMAssay Description:Displacement of [3H]CP55490 from human recombinant cannabinoid CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323608(CHEMBL1209597 | rac-(S)-N-(3-(3-bromophenyl)-4-(4-...)
Affinity DataIC50:  22nMAssay Description:Displacement of [3H]CP55490 from human recombinant cannabinoid CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323610(CHEMBL1209668 | N-(3-(3-bromophenyl)-4-(4-chloroph...)
Affinity DataIC50:  25nMAssay Description:Displacement of [3H]CP55490 from human recombinant cannabinoid CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323610(CHEMBL1209668 | N-(3-(3-bromophenyl)-4-(4-chloroph...)
Affinity DataIC50:  25nMAssay Description:Displacement of [3H]CP55490 from human recombinant cannabinoid CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323609((+/-)-N-(2-(3-bromophenyl)-3-(4-chlorophenyl)-2-me...)
Affinity DataIC50:  340nMAssay Description:Displacement of [3H]CP55490 from human recombinant cannabinoid CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323612((+/-)-1-(3-(4-chlorobenzyl)-3-phenylpyrrolidin-1-y...)
Affinity DataIC50:  810nMAssay Description:Displacement of [3H]CP55490 from human recombinant cannabinoid CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323611((+/-)-1-(3-(4-chlorobenzyl)-3-phenylazetidin-1-yl)...)
Affinity DataIC50:  1.30E+3nMAssay Description:Displacement of [3H]CP55490 from human recombinant cannabinoid CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50323613((+/-)-1-(3-(4-chlorobenzyl)-3-phenylpiperidin-1-yl...)
Affinity DataIC50:  2.00E+3nMAssay Description:Displacement of [3H]CP55490 from human recombinant cannabinoid CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed