Compile Data Set for Download or QSAR
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Found 13 Enz. Inhib. hit(s) with all data for entry = 50032512
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034839(8-Chloro-5-methyl-6-oxo-5,6-dihydro-4H-2,5,10b-tri...)
Affinity DataKi:  6.80nMAssay Description:Binding affinity to human recombinant GABA alpha1beta2gamma2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
University Of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034839(8-Chloro-5-methyl-6-oxo-5,6-dihydro-4H-2,5,10b-tri...)
Affinity DataKi:  9.20nMAssay Description:Binding affinity to human recombinant GABA alpha3beta2gamma2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Homo sapiens (Human))
University Of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034839(8-Chloro-5-methyl-6-oxo-5,6-dihydro-4H-2,5,10b-tri...)
Affinity DataKi:  16.3nMAssay Description:Binding affinity to human recombinant GABA alpha2beta2gamma2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA A receptor alpha-4/beta-3/gamma-2(Homo sapiens (Human))
University Of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034820(8-Chloro-3-methoxymethyl-5-methyl-4,5-dihydro-2,5,...)
Affinity DataKi:  38.8nMAssay Description:Binding affinity to human recombinant GABA alpha4beta3gamma2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))
University Of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034820(8-Chloro-3-methoxymethyl-5-methyl-4,5-dihydro-2,5,...)
Affinity DataKi: >300nMAssay Description:Binding affinity to human recombinant GABA alpha2beta3gamma2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
University Of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034820(8-Chloro-3-methoxymethyl-5-methyl-4,5-dihydro-2,5,...)
Affinity DataKi: >300nMAssay Description:Binding affinity to human recombinant GABA alpha5beta3gamma2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
University Of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034820(8-Chloro-3-methoxymethyl-5-methyl-4,5-dihydro-2,5,...)
Affinity DataKi: >300nMAssay Description:Binding affinity to human recombinant GABA alpha1beta3gamma2 receptorMore data for this Ligand-Target Pair
Target InfoGoogleScholar
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Homo sapiens (Human))
University Of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034820(8-Chloro-3-methoxymethyl-5-methyl-4,5-dihydro-2,5,...)
Affinity DataKi: >300nMAssay Description:Binding affinity to human recombinant GABA alpha3beta3gamma2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA A receptor alpha-4/beta-3/gamma-2(Homo sapiens (Human))
University Of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034826(3-Acetyl-8-chloro-5-methyl-4,5-dihydro-2,5,10b-tri...)
Affinity DataKi:  2.61E+3nMAssay Description:Binding affinity to human recombinant GABA alpha4beta3gamma2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
University Of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034826(3-Acetyl-8-chloro-5-methyl-4,5-dihydro-2,5,10b-tri...)
Affinity DataKi:  1.75E+4nMAssay Description:Binding affinity to human recombinant GABA alpha1beta3gamma2 receptorMore data for this Ligand-Target Pair
Target InfoGoogleScholar
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Homo sapiens (Human))
University Of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034826(3-Acetyl-8-chloro-5-methyl-4,5-dihydro-2,5,10b-tri...)
Affinity DataKi:  2.21E+4nMAssay Description:Binding affinity to human recombinant GABA alpha3beta3gamma2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
University Of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034826(3-Acetyl-8-chloro-5-methyl-4,5-dihydro-2,5,10b-tri...)
Affinity DataKi:  2.95E+4nMAssay Description:Binding affinity to human recombinant GABA alpha5beta3gamma2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))
University Of Massachusetts

Curated by ChEMBL
LigandPNGBDBM50034826(3-Acetyl-8-chloro-5-methyl-4,5-dihydro-2,5,10b-tri...)
Affinity DataKi:  3.38E+4nMAssay Description:Binding affinity to human recombinant GABA alpha2beta3gamma2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed