Compile Data Set for Download or QSAR
maximum 50k data
Found 52 Enz. Inhib. hit(s) with all data for entry = 50032152
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50202986(2-furan-2-yl-7-(2-{4-[4-(2-methoxy-ethoxy)-phenyl]...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324983(CHEMBL1221457 | Cyclopropanecarboxylic acid[5-(3-m...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324967(2-[(Furan-2-carbonyl)-amino]-4-phenyl-thiazole-5-c...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324975(CHEMBL1222306 | N-[5-(5-Methyl-[1,2,4]oxadiazol-3-...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324984(3-Methyl-N-[5-(3-methyl-[1,2,4]oxadiazol-5-yl)-4-p...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324972(CHEMBL1222303 | Cyclopropanecarboxylic acid[5-(5-m...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324973(3-Methyl-N-[5-(5-methyl-[1,2,4]oxadiazol-3-yl)-4-p...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324983(CHEMBL1221457 | Cyclopropanecarboxylic acid[5-(3-m...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324991(2-(3,4-Dimethoxy-phenyl)-N-[5-(2-ethyl-2H-tetrazol...)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324984(3-Methyl-N-[5-(3-methyl-[1,2,4]oxadiazol-5-yl)-4-p...)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324986(CHEMBL1221504 | N-[5-(3-Methyl-[1,2,4]oxadiazol-5-...)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324968(CHEMBL1222241 | Furan-2-carboxylic acid(5-butyryl-...)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50176050(8-(3,4-dimethoxystyryl)-1,3-diethyl-7-methyl-1H-pu...)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324988(CHEMBL1221506 | Cyclopropanecarboxylic acid[5-(2-e...)
Affinity DataKi:  77nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324978(3-Methyl-N-(5-[1,2,4]oxadiazol-3-yl-4-phenyl-thiaz...)
Affinity DataKi:  77nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324973(3-Methyl-N-[5-(5-methyl-[1,2,4]oxadiazol-3-yl)-4-p...)
Affinity DataKi:  82nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324974(CHEMBL1222305 | N-[5-(5-Methyl-[1,2,4]oxadiazol-3-...)
Affinity DataKi:  83nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324968(CHEMBL1222241 | Furan-2-carboxylic acid(5-butyryl-...)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324969(CHEMBL1222242 | Furan-2-carboxylic acid(5-ethoxyme...)
Affinity DataKi:  92nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324987(CHEMBL1221505 | Furan-2-carboxylic acid[5-(2-ethyl...)
Affinity DataKi:  94nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324967(2-[(Furan-2-carbonyl)-amino]-4-phenyl-thiazole-5-c...)
Affinity DataKi:  95nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324982(CHEMBL1221456 | N-[5-(3-Methyl-[1,2,4]oxadiazol-5-...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324977(CHEMBL1222370 | Cyclopropanecarboxylic acid(5-[1,2...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324972(CHEMBL1222303 | Cyclopropanecarboxylic acid[5-(5-m...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324985(CHEMBL1221459 | N-[5-(3-Methyl-[1,2,4]oxadiazol-5-...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324969(CHEMBL1222242 | Furan-2-carboxylic acid(5-ethoxyme...)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324985(CHEMBL1221459 | N-[5-(3-Methyl-[1,2,4]oxadiazol-5-...)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324971(CHEMBL1222302 | N-[5-(5-Methyl-[1,2,4]oxadiazol-3-...)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324981(CHEMBL1221455 | Furan-2-carboxylic acid[5-(3-methy...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324988(CHEMBL1221506 | Cyclopropanecarboxylic acid[5-(2-e...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324989(CHEMBL1221507 | N-[5-(2-Ethyl-2H-tetrazol-5-yl)-4-...)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324976(CHEMBL1222369 | Furan-2-carboxylic acid(5-[1,2,4]o...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324975(CHEMBL1222306 | N-[5-(5-Methyl-[1,2,4]oxadiazol-3-...)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324981(CHEMBL1221455 | Furan-2-carboxylic acid[5-(3-methy...)
Affinity DataKi:  270nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324992(CHEMBL1222245 | Furan-2-carboxylic acid(5-cyano-4-...)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324979(CHEMBL1222372 | N-(5-[1,2,4]Oxadiazol-3-yl-4-pheny...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324977(CHEMBL1222370 | Cyclopropanecarboxylic acid(5-[1,2...)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324979(CHEMBL1222372 | N-(5-[1,2,4]Oxadiazol-3-yl-4-pheny...)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324978(3-Methyl-N-(5-[1,2,4]oxadiazol-3-yl-4-phenyl-thiaz...)
Affinity DataKi:  340nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324986(CHEMBL1221504 | N-[5-(3-Methyl-[1,2,4]oxadiazol-5-...)
Affinity DataKi:  340nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324982(CHEMBL1221456 | N-[5-(3-Methyl-[1,2,4]oxadiazol-5-...)
Affinity DataKi:  370nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324976(CHEMBL1222369 | Furan-2-carboxylic acid(5-[1,2,4]o...)
Affinity DataKi:  410nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324990(CHEMBL1221508 | N-[5-(2-Ethyl-2H-tetrazol-5-yl)-4-...)
Affinity DataKi:  460nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324987(CHEMBL1221505 | Furan-2-carboxylic acid[5-(2-ethyl...)
Affinity DataKi:  650nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324970(CHEMBL1222246 | Furan-2-carboxylic acid[5-(5-methy...)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324980(CHEMBL1222373 | N-(5-[1,2,4]Oxadiazol-3-yl-4-pheny...)
Affinity DataKi:  710nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324970(CHEMBL1222246 | Furan-2-carboxylic acid[5-(5-methy...)
Affinity DataKi:  780nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50202986(2-furan-2-yl-7-(2-{4-[4-(2-methoxy-ethoxy)-phenyl]...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324990(CHEMBL1221508 | N-[5-(2-Ethyl-2H-tetrazol-5-yl)-4-...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324991(2-(3,4-Dimethoxy-phenyl)-N-[5-(2-ethyl-2H-tetrazol...)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 52 total ) | Next | Last >>
Jump to: