Compile Data Set for Download or QSAR
maximum 50k data
Found 40 Enz. Inhib. hit(s) with all data for entry = 50039270
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  1.60nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST4 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  2.30nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST1 receptor expressed in CHO cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  2.40nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST5 receptor expressed in HEK293 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST2 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50159392((4R,7R,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-37...)
Affinity DataIC50:  3.60nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST3 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325031(4-(((3S,6S,9R,12S,15S,20S,Z)-9-((1H-indol-2-yl)met...)
Affinity DataIC50:  4.90nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST5 receptor expressed in HEK293 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325028((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50:  9.60nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST2 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325027(4-(((3S,6S,9R,12S,15S,20S,Z)-9-((1H-indol-2-yl)met...)
Affinity DataIC50:  12.3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST5 receptor expressed in HEK293 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325028((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50:  16.5nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST5 receptor expressed in HEK293 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325027(4-(((3S,6S,9R,12S,15S,20S,Z)-9-((1H-indol-2-yl)met...)
Affinity DataIC50:  25nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST1 receptor expressed in CHO cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325027(4-(((3S,6S,9R,12S,15S,20S,Z)-9-((1H-indol-2-yl)met...)
Affinity DataIC50:  25nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST3 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325033((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50:  28nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST5 receptor expressed in HEK293 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325034(4-(((3S,6S,9R,12S,15S,20S,E)-9-((1H-indol-2-yl)met...)
Affinity DataIC50:  29nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST5 receptor expressed in HEK293 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325033((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50:  44nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST2 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325027(4-(((3S,6S,9R,12S,15S,20S,Z)-9-((1H-indol-2-yl)met...)
Affinity DataIC50:  46nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST2 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325031(4-(((3S,6S,9R,12S,15S,20S,Z)-9-((1H-indol-2-yl)met...)
Affinity DataIC50:  57.5nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST1 receptor expressed in CHO cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325030((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50:  87nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST2 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325031(4-(((3S,6S,9R,12S,15S,20S,Z)-9-((1H-indol-2-yl)met...)
Affinity DataIC50:  92.5nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST3 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325031(4-(((3S,6S,9R,12S,15S,20S,Z)-9-((1H-indol-2-yl)met...)
Affinity DataIC50:  101nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST2 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325030((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50:  161nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST5 receptor expressed in HEK293 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325028((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50:  249nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST4 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325027(4-(((3S,6S,9R,12S,15S,20S,Z)-9-((1H-indol-2-yl)met...)
Affinity DataIC50:  346nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST4 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325029((2S,5R,8S,11S,14S,19S,E)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50:  356nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST2 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325033((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50:  412nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST4 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325029((2S,5R,8S,11S,14S,19S,E)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50:  418nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST5 receptor expressed in HEK293 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325034(4-(((3S,6S,9R,12S,15S,20S,E)-9-((1H-indol-2-yl)met...)
Affinity DataIC50:  892nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST3 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325033((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST1 receptor expressed in CHO cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325028((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST1 receptor expressed in CHO cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325029((2S,5R,8S,11S,14S,19S,E)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST1 receptor expressed in CHO cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325030((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST1 receptor expressed in CHO cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325029((2S,5R,8S,11S,14S,19S,E)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST3 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325028((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST3 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325034(4-(((3S,6S,9R,12S,15S,20S,E)-9-((1H-indol-2-yl)met...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST2 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325033((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST3 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325029((2S,5R,8S,11S,14S,19S,E)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST4 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325034(4-(((3S,6S,9R,12S,15S,20S,E)-9-((1H-indol-2-yl)met...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST4 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325031(4-(((3S,6S,9R,12S,15S,20S,Z)-9-((1H-indol-2-yl)met...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST4 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325030((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST4 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325034(4-(((3S,6S,9R,12S,15S,20S,E)-9-((1H-indol-2-yl)met...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST1 receptor expressed in CHO cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Firenze

Curated by ChEMBL
LigandPNGBDBM50325030((2S,5R,8S,11S,14S,19S,Z)-5-((1H-indol-2-yl)methyl)...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-[LTT] SIRF-28 from human SST3 receptor expressed in human CCL39 cells by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed