Affinity DataKi: 0.631nMAssay Description:Antagonist activity at human recombinant histamine H1 receptor expressed in CHO cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.16nMAssay Description:Antagonist activity at human adrenergic Alpha-1B receptor assessed as intracellular calcium luminescence by cell based aequorin assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.98nMAssay Description:Antagonist activity at human adrenergic alpha1A receptor assessed as intracellular calcium luminescence by cell based aequorin assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.94nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in HEK cells assessed as intracellular calcium luminescence by aequorin assayMore data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:Antagonist activity at human recombinant histamine H1 receptor expressed in CHO cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:Antagonist activity at human recombinant histamine H1 receptor expressed in CHO cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 15.8nMAssay Description:Antagonist activity at human 5HT2B receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 19.9nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 19.9nMAssay Description:Antagonist activity at human recombinant histamine H1 receptor expressed in CHO cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 25.1nMAssay Description:Antagonist activity at human 5HT2B receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 25.1nMAssay Description:Antagonist activity at human recombinant histamine H1 receptor expressed in CHO cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 31.6nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 31.6nMAssay Description:Antagonist activity at human recombinant histamine H1 receptor expressed in CHO cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 39.8nMAssay Description:Antagonist activity at human 5HT2B receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 39.8nMAssay Description:Antagonist activity at human 5HT2B receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 39.8nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in HEK cells assessed as intracellular calcium luminescence by aequorin assayMore data for this Ligand-Target Pair
Affinity DataKi: 39.8nMAssay Description:Antagonist activity at human recombinant histamine H1 receptor expressed in CHO cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 39.8nMAssay Description:Antagonist activity at human recombinant histamine H1 receptor expressed in CHO cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 39.8nMAssay Description:Antagonist activity at human recombinant histamine H1 receptor expressed in CHO cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 50.1nMAssay Description:Antagonist activity at human recombinant histamine H1 receptor expressed in CHO cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 50.1nMAssay Description:Antagonist activity at human recombinant histamine H1 receptor expressed in CHO cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 50.1nMAssay Description:Antagonist activity at human recombinant histamine H1 receptor expressed in CHO cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 50.1nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 50.1nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in HEK cells assessed as intracellular calcium luminescence by aequorin assayMore data for this Ligand-Target Pair
Affinity DataKi: 63.1nMAssay Description:Antagonist activity at human 5HT2B receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 63.1nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in HEK cells assessed as intracellular calcium luminescence by aequorin assayMore data for this Ligand-Target Pair
Affinity DataKi: 63.1nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 79.4nMAssay Description:Antagonist activity at human recombinant histamine H1 receptor expressed in CHO cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 79.4nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in HEK cells assessed as intracellular calcium luminescence by aequorin assayMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Antagonist activity at human 5HT2B receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in HEK cells assessed as intracellular calcium luminescence by aequorin assayMore data for this Ligand-Target Pair
Affinity DataKi: 125nMAssay Description:Antagonist activity at human recombinant histamine H1 receptor expressed in CHO cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Antagonist activity at human recombinant histamine H1 receptor expressed in CHO cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Antagonist activity at human recombinant histamine H1 receptor expressed in CHO cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in HEK cells assessed as intracellular calcium luminescence by aequorin assayMore data for this Ligand-Target Pair
Affinity DataKi: 158nMAssay Description:Antagonist activity at human 5HT2B receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 158nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in HEK cells assessed as intracellular calcium luminescence by aequorin assayMore data for this Ligand-Target Pair
Affinity DataKi: 251nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in HEK cells assessed as intracellular calcium luminescence by aequorin assayMore data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in HEK cells assessed as intracellular calcium luminescence by aequorin assayMore data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Antagonist activity at human 5HT2B receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Antagonist activity at human 5HT2B receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 398nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in HEK cells assessed as intracellular calcium luminescence by aequorin assayMore data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 630nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in HEK cells assessed as intracellular calcium luminescence by aequorin assayMore data for this Ligand-Target Pair
Affinity DataKi: 631nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in HEK cells assessed as intracellular calcium luminescence by aequorin assayMore data for this Ligand-Target Pair