Compile Data Set for Download or QSAR
maximum 50k data
Found 41 Enz. Inhib. hit(s) with all data for entry = 50032185
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(CHEMBL1224034 | N-cyclohexyl-8-fluoro-3,3a,4,9b-te...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325659(8-fluoro-N-phenyl-3,3a,4,9b-tetrahydro-1H-thiochro...)
Affinity DataKi:  223nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325661(8-fluoro-N-propyl-3,3a,4,9b-tetrahydro-1H-thiochro...)
Affinity DataKi:  384nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325663(CHEMBL1224035 | N-butyl-8-fluoro-3,3a,4,9b-tetrahy...)
Affinity DataKi:  489nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325660(8-fluoro-N-isopropyl-3,3a,4,9b-tetrahydro-1H-thioc...)
Affinity DataKi:  569nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325664(CHEMBL1224036 | N-phenyl-3,3a,4,9b-tetrahydro-1H-c...)
Affinity DataKi:  1.61E+3nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325667(CHEMBL1224103 | N-cyclohexyl-3,3a,4,9b-tetrahydro-...)
Affinity DataKi:  1.77E+3nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325670(CHEMBL1224106 | N-o-tolyl-3,3a,4,9b-tetrahydro-1H-...)
Affinity DataKi:  4.00E+3nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325659(8-fluoro-N-phenyl-3,3a,4,9b-tetrahydro-1H-thiochro...)
Affinity DataKi:  5.17E+3nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325666(CHEMBL1224102 | N-propyl-3,3a,4,9b-tetrahydro-1H-c...)
Affinity DataKi:  6.60E+3nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325664(CHEMBL1224036 | N-phenyl-3,3a,4,9b-tetrahydro-1H-c...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325665(CHEMBL1224101 | N-isopropyl-3,3a,4,9b-tetrahydro-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325665(CHEMBL1224101 | N-isopropyl-3,3a,4,9b-tetrahydro-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325666(CHEMBL1224102 | N-propyl-3,3a,4,9b-tetrahydro-1H-c...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325666(CHEMBL1224102 | N-propyl-3,3a,4,9b-tetrahydro-1H-c...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325667(CHEMBL1224103 | N-cyclohexyl-3,3a,4,9b-tetrahydro-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325667(CHEMBL1224103 | N-cyclohexyl-3,3a,4,9b-tetrahydro-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325668(CHEMBL1224104 | N-tert-butyl-3,3a,4,9b-tetrahydro-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325668(CHEMBL1224104 | N-tert-butyl-3,3a,4,9b-tetrahydro-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325668(CHEMBL1224104 | N-tert-butyl-3,3a,4,9b-tetrahydro-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325669(CHEMBL1224105 | N-butyl-3,3a,4,9b-tetrahydro-1H-ch...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325669(CHEMBL1224105 | N-butyl-3,3a,4,9b-tetrahydro-1H-ch...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325669(CHEMBL1224105 | N-butyl-3,3a,4,9b-tetrahydro-1H-ch...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325670(CHEMBL1224106 | N-o-tolyl-3,3a,4,9b-tetrahydro-1H-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325664(CHEMBL1224036 | N-phenyl-3,3a,4,9b-tetrahydro-1H-c...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325663(CHEMBL1224035 | N-butyl-8-fluoro-3,3a,4,9b-tetrahy...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325663(CHEMBL1224035 | N-butyl-8-fluoro-3,3a,4,9b-tetrahy...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(CHEMBL1224034 | N-cyclohexyl-8-fluoro-3,3a,4,9b-te...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(CHEMBL1224034 | N-cyclohexyl-8-fluoro-3,3a,4,9b-te...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325661(8-fluoro-N-propyl-3,3a,4,9b-tetrahydro-1H-thiochro...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325661(8-fluoro-N-propyl-3,3a,4,9b-tetrahydro-1H-thiochro...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325660(8-fluoro-N-isopropyl-3,3a,4,9b-tetrahydro-1H-thioc...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325660(8-fluoro-N-isopropyl-3,3a,4,9b-tetrahydro-1H-thioc...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325659(8-fluoro-N-phenyl-3,3a,4,9b-tetrahydro-1H-thiochro...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325665(CHEMBL1224101 | N-isopropyl-3,3a,4,9b-tetrahydro-1...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(CHEMBL1224034 | N-cyclohexyl-8-fluoro-3,3a,4,9b-te...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Citalopram from human SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325670(CHEMBL1224106 | N-o-tolyl-3,3a,4,9b-tetrahydro-1H-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(CHEMBL1224034 | N-cyclohexyl-8-fluoro-3,3a,4,9b-te...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]WIN-3542 from human DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(CHEMBL1224034 | N-cyclohexyl-8-fluoro-3,3a,4,9b-te...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Nisoxetine from human NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(CHEMBL1224034 | N-cyclohexyl-8-fluoro-3,3a,4,9b-te...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human 5HT2B receptor assessed as 10633-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Csiro Molecular And Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(CHEMBL1224034 | N-cyclohexyl-8-fluoro-3,3a,4,9b-te...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human 5HT2C receptor assessed as 10633-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed