Compile Data Set for Download or QSAR
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Found 58 Enz. Inhib. hit(s) with all data for entry = 50041865
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417295(CHEMBL1276325)
Affinity DataIC50:  0.288nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417313(CHEMBL1276585)
Affinity DataIC50:  0.501nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50026568(CHEMBL23464 | N-(1-Ethyl-pyrrolidin-2-ylmethyl)-3-...)
Affinity DataIC50:  0.676nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417312(CHEMBL1276560)
Affinity DataIC50:  0.912nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417296(CHEMBL1276326)
Affinity DataIC50:  1.10nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50026045((R,S)-3-Bromo-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2,...)
Affinity DataIC50:  1.20nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50026565(3-Ethyl-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2,6-dime...)
Affinity DataIC50:  1.29nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417297(CHEMBL1276327)
Affinity DataIC50:  1.29nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417307(CHEMBL1276494)
Affinity DataIC50:  1.41nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417311(CHEMBL1276559)
Affinity DataIC50:  1.51nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417320(CHEMBL1276712)
Affinity DataIC50:  1.70nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417335(CHEMBL1276647)
Affinity DataIC50:  1.78nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417332(CHEMBL1276561)
Affinity DataIC50:  2.29nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417298(CHEMBL1276350)
Affinity DataIC50:  2.69nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417331(CHEMBL1276529)
Affinity DataIC50:  2.88nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417330(CHEMBL1276496)
Affinity DataIC50:  3.02nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417315(CHEMBL1276615)
Affinity DataIC50:  3.24nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417301(CHEMBL1276375)
Affinity DataIC50:  4.17nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417292(CHEMBL1276763)
Affinity DataIC50:  5.01nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417316(CHEMBL1276645)
Affinity DataIC50:  5.25nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417334(CHEMBL1276616)
Affinity DataIC50:  5.5nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417300(CHEMBL1276374)
Affinity DataIC50:  5.62nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417338(CHEMBL1276740)
Affinity DataIC50:  7.08nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417310(CHEMBL1276528)
Affinity DataIC50:  7.76nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417290(CHEMBL1276738)
Affinity DataIC50:  7.94nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417328(CHEMBL1276459)
Affinity DataIC50:  8.32nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417302(CHEMBL1276400)
Affinity DataIC50:  8.71nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50007534(3-Bromo-N-((S)-1-ethyl-pyrrolidin-2-ylmethyl)-2-hy...)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417319(CHEMBL1276711)
Affinity DataIC50:  11.0nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417291(CHEMBL1276739)
Affinity DataIC50:  11.0nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417321(CHEMBL1276741)
Affinity DataIC50:  11.0nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417305(CHEMBL1276428)
Affinity DataIC50:  12.0nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417317(CHEMBL1276646)
Affinity DataIC50:  17.0nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417306(CHEMBL1276460)
Affinity DataIC50:  17.0nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417322(CHEMBL1276742)
Affinity DataIC50:  19.1nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417299(CHEMBL1276352)
Affinity DataIC50:  19.9nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417329(CHEMBL1276461)
Affinity DataIC50:  25.7nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417309(CHEMBL1276527)
Affinity DataIC50:  25.7nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417288(CHEMBL1276708)
Affinity DataIC50:  32.4nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417327(CHEMBL1276426)
Affinity DataIC50:  38.9nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417336(CHEMBL1276677)
Affinity DataIC50:  39.8nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417325(CHEMBL1276268)
Affinity DataIC50:  45.7nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50026566(CHEMBL282024 | N-(1-Ethyl-pyrrolidin-2-ylmethyl)-2...)
Affinity DataIC50:  52.5nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417337(CHEMBL1276710)
Affinity DataIC50:  56.2nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417304(CHEMBL1276427)
Affinity DataIC50:  57.5nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417326(CHEMBL1276399)
Affinity DataIC50:  64.6nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417340(CHEMBL1276351)
Affinity DataIC50:  67.6nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417333(CHEMBL1276587)
Affinity DataIC50:  67.6nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417289(CHEMBL1276709)
Affinity DataIC50:  70.8nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Mazandaran

Curated by ChEMBL
LigandPNGBDBM50417293(CHEMBL1276764)
Affinity DataIC50:  110nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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