Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50033224
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita` Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50341606(1-(2,5-dimethoxyphenyl)-3-(4-oxo-3-phenyl-3,4-dihy...)
Affinity DataKi:  0.776nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita` Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50341605(4-(2-Methoxyphenyl)ureido-2-phenylphthalazin-1(2H)...)
Affinity DataKi:  8.90nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita` Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50341604(1-(3-methoxyphenyl)-3-(4-oxo-3-phenyl-3,4-dihydrop...)
Affinity DataKi:  9.75nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita` Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50341607(1-benzyl-3-(4-oxo-3-phenyl-3,4-dihydrophthalazin-1...)
Affinity DataKi:  29.6nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Universita` Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50086145(1-(1-Oxo-2-phenyl-1,2-dihydro-[1,2,4]triazolo[4,3-...)
Affinity DataKi:  50.8nMAssay Description:Displacement of [3H]CHA from adenosine A1 receptor in bovine brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita` Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50341603(1-(4-methoxyphenyl)-3-(4-oxo-3-phenyl-3,4-dihydrop...)
Affinity DataKi:  60.6nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita` Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50341602(1-(4-oxo-3-phenyl-3,4-dihydrophthalazin-1-yl)-3-ph...)
Affinity DataKi:  178nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita` Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50341608(1-(2-methoxybenzyl)-3-(4-oxo-3-phenyl-3,4-dihydrop...)
Affinity DataKi:  274nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita` Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50086145(1-(1-Oxo-2-phenyl-1,2-dihydro-[1,2,4]triazolo[4,3-...)
Affinity DataKi:  276nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita` Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50086153(4-Amino-2-phenyl-2H-[1,2,4]triazolo[4,3-a]quinoxal...)
Affinity DataKi:  490nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita` Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50341601(CHEMBL1766267 | N-(4-oxo-3-phenyl-3,4-dihydrophtha...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita` Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50341607(1-benzyl-3-(4-oxo-3-phenyl-3,4-dihydrophthalazin-1...)
Affinity DataIC50:  1.15nMAssay Description:Antagonist activity at human cloned adenosine A3 receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP accumulation after 15 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita` Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50341606(1-(2,5-dimethoxyphenyl)-3-(4-oxo-3-phenyl-3,4-dihy...)
Affinity DataIC50:  8.25nMAssay Description:Antagonist activity at human cloned adenosine A3 receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP accumulation after 15 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita` Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50341605(4-(2-Methoxyphenyl)ureido-2-phenylphthalazin-1(2H)...)
Affinity DataIC50:  17nMAssay Description:Antagonist activity at human cloned adenosine A3 receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP accumulation after 15 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita` Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50341604(1-(3-methoxyphenyl)-3-(4-oxo-3-phenyl-3,4-dihydrop...)
Affinity DataIC50:  18nMAssay Description:Antagonist activity at human cloned adenosine A3 receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP accumulation after 15 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita` Degli Studi Di Firenze

Curated by ChEMBL
LigandPNGBDBM50341603(1-(4-methoxyphenyl)-3-(4-oxo-3-phenyl-3,4-dihydrop...)
Affinity DataIC50:  28nMAssay Description:Antagonist activity at human cloned adenosine A3 receptor expressed in CHO cells assessed as inhibition of NECA-induced cAMP accumulation after 15 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed