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Found 5 Enz. Inhib. hit(s) with all data for entry = 50033151
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50340427(1-((3S,8S,9S,10R,13S,14S,17R)-16-(benzylamino)-3-h...)
Affinity DataIC50:  2.13E+4nMAssay Description:Inhibition of human DPP-4 assessed as cleavage of substrate using H-Gly-Pro-AMC chromogenic substrate after 10 mins by double beam spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50340428(3-(3,4-dimethoxyphenyl)-1-((3S,8R,9S,10R,13S,14S)-...)
Affinity DataIC50:  2.62E+4nMAssay Description:Inhibition of human DPP-4 assessed as cleavage of substrate using H-Gly-Pro-AMC chromogenic substrate after 10 mins by double beam spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50340430((2S,4aR,4bS,6aS,9R,11aS,11bS)-2-Hydroxy-9-(4-isopr...)
Affinity DataIC50:  2.91E+4nMAssay Description:Inhibition of human DPP-4 assessed as cleavage of substrate using H-Gly-Pro-AMC chromogenic substrate after 10 mins by double beam spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50340429((2S,4aR,4bS,6aS,9R,11aS,11bS)-2-Hydroxy-9-(4-metho...)
Affinity DataIC50:  3.27E+4nMAssay Description:Inhibition of human DPP-4 assessed as cleavage of substrate using H-Gly-Pro-AMC chromogenic substrate after 10 mins by double beam spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50340426(16-Dehydropregnenolone acetate | CHEMBL1761683)
Affinity DataIC50:  3.56E+4nMAssay Description:Inhibition of human DPP-4 assessed as cleavage of substrate using H-Gly-Pro-AMC chromogenic substrate after 10 mins by double beam spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed