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Found 29 Enz. Inhib. hit(s) with all data for entry = 50034083
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50156916((1R)-3beta-(4-bromophenyl)tropane-2beta-carboxylic...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [125I]-IPT from DAT transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356626(CHEMBL1914699)
Affinity DataKi:  4.10nMAssay Description:Displacement of [125I]-IPT from DAT transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50304045(CHEMBL608703 | methyl 3-(4-chlorophenyl)-8-methyl-...)
Affinity DataKi:  5.10nMAssay Description:Displacement of [125I]-IPT from DAT transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356629(CHEMBL1914696)
Affinity DataKi:  5.60nMAssay Description:Displacement of [125I]-IPT from DAT transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356629(CHEMBL1914696)
Affinity DataKi:  7.40nMAssay Description:Displacement of [125I]-IDAM from SERT transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356627(CHEMBL1914698)
Affinity DataKi:  7.90nMAssay Description:Displacement of [125I]-IPT from DAT transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356627(CHEMBL1914698)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]-IDAM from SERT transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356628(CHEMBL1914697)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]-IDAM from SERT transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50451132(CHEMBL2079586 | WIN-35428)
Affinity DataKi:  15nMAssay Description:Displacement of [125I]-IPT from DAT transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356628(CHEMBL1914697)
Affinity DataKi:  18nMAssay Description:Displacement of [125I]-IPT from DAT transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356626(CHEMBL1914699)
Affinity DataKi:  21nMAssay Description:Displacement of [125I]-IDAM from SERT transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356627(CHEMBL1914698)
Affinity DataKi:  28nMAssay Description:Displacement of [125I]-INXT from NET transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356629(CHEMBL1914696)
Affinity DataKi:  29nMAssay Description:Displacement of [125I]-INXT from NET transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356628(CHEMBL1914697)
Affinity DataKi:  49nMAssay Description:Displacement of [125I]-INXT from NET transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356626(CHEMBL1914699)
Affinity DataKi:  66nMAssay Description:Displacement of [125I]-INXT from NET transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356631(CHEMBL1914694)
Affinity DataKi:  82nMAssay Description:Displacement of [125I]-IPT from DAT transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356633(CHEMBL1914692)
Affinity DataKi:  87nMAssay Description:Displacement of [125I]-IPT from DAT transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356632(CHEMBL1914693)
Affinity DataKi:  106nMAssay Description:Displacement of [125I]-IPT from DAT transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356630(CHEMBL1914695)
Affinity DataKi:  127nMAssay Description:Displacement of [125I]-IPT from DAT transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50451132(CHEMBL2079586 | WIN-35428)
Affinity DataKi:  181nMAssay Description:Displacement of [125I]-IDAM from SERT transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50451132(CHEMBL2079586 | WIN-35428)
Affinity DataKi:  635nMAssay Description:Displacement of [125I]-INXT from NET transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356633(CHEMBL1914692)
Affinity DataKi:  3.21E+3nMAssay Description:Displacement of [125I]-IDAM from SERT transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356633(CHEMBL1914692)
Affinity DataKi:  3.86E+3nMAssay Description:Displacement of [125I]-INXT from NET transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356631(CHEMBL1914694)
Affinity DataKi:  1.03E+4nMAssay Description:Displacement of [125I]-IDAM from SERT transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356631(CHEMBL1914694)
Affinity DataKi:  1.21E+4nMAssay Description:Displacement of [125I]-INXT from NET transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356632(CHEMBL1914693)
Affinity DataKi:  1.53E+4nMAssay Description:Displacement of [125I]-IDAM from SERT transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356632(CHEMBL1914693)
Affinity DataKi:  1.62E+4nMAssay Description:Displacement of [125I]-INXT from NET transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356630(CHEMBL1914695)
Affinity DataKi:  1.69E+4nMAssay Description:Displacement of [125I]-INXT from NET transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Key Laboratory Of Radiopharmaceuticals (Beijing Normal University)

Curated by ChEMBL
LigandPNGBDBM50356630(CHEMBL1914695)
Affinity DataKi:  2.91E+4nMAssay Description:Displacement of [125I]-IDAM from SERT transfected in pig LLC-PK1 cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed