Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 50033430
TargetAromatase(Homo sapiens (Human))
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM13061(4,4 -(1H-1,2,4-triazol-1-ylmethanediyl)dibenzonitr...)
Affinity DataIC50:  18nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAromatase(Homo sapiens (Human))
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50345191(7,8-Benzo-4'-hydroxy-4-imidazolylflavan | CHEMBL17...)
Affinity DataIC50:  32nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50345190(2,4-cis-7,8-benzo-4'-cyano-4-imidazolylflavan | 2,...)
Affinity DataIC50:  34nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50345189(2,4-trans-7,8-benzo-4-imidazolylflavan | CHEMBL178...)
Affinity DataIC50:  36nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50118966(1-(7-Methoxy-2-phenyl-chroman-4-yl)-1H-imidazole |...)
Affinity DataIC50:  60nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50118966(1-(7-Methoxy-2-phenyl-chroman-4-yl)-1H-imidazole |...)
Affinity DataIC50:  91nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50118966(1-(7-Methoxy-2-phenyl-chroman-4-yl)-1H-imidazole |...)
Affinity DataIC50:  91nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50345190(2,4-cis-7,8-benzo-4'-cyano-4-imidazolylflavan | 2,...)
Affinity DataIC50:  534nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50345190(2,4-cis-7,8-benzo-4'-cyano-4-imidazolylflavan | 2,...)
Affinity DataIC50:  534nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50345188(2-(4-hydroxyphenyl)-2,3-dihydrobenzo[h]chromen-4-o...)
Affinity DataIC50:  630nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50345187(4-(4-oxo-3,4-dihydro-2H-benzo[h]chromen-2-yl)benzo...)
Affinity DataIC50:  1.54E+3nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50345186(2-phenyl-2,3-dihydrobenzo[h]chromen-4-one | 2-phen...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM9460(3-(4-aminophenyl)-3-ethyl-piperidine-2,6-dione | 3...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank