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Found 28 Enz. Inhib. hit(s) with all data for entry = 50033410
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50293015(CHEMBL502503 | Methyl 4-((4-(2-(6,7-Dimethoxy-1,2,...)
Affinity DataIC50:  59nMAssay Description:Inhibition of ABCG2 expressed in human MCF7/Topo cells by Hoechst microplate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50206310(5-Methoxy-9-oxo-9,10-dihydro-acridine-4-carboxylic...)
Affinity DataIC50:  127nMAssay Description:Inhibition of ABCG2 expressed in human MCF7/Topo cells by Hoechst microplate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50344753(CHEMBL1779526 | N-{4-[2-(6-Methoxy-7-{2-[2-(2-meth...)
Affinity DataIC50:  130nMAssay Description:Inhibition of ABCG2 expressed in human MCF7/Topo cells by Hoechst microplate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50293013(CHEMBL455275 | Methyl 4-((4-(2-(6,7-dimethoxy-1,2,...)
Affinity DataIC50:  172nMAssay Description:Inhibition of ABCG2 expressed in human MCF7/Topo cells by Hoechst microplate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50344755(CHEMBL1779524 | N-{4-[2-(7-Methoxy-6-{2-[2-(2-meth...)
Affinity DataIC50:  183nMAssay Description:Inhibition of ABCG2 expressed in human MCF7/Topo cells by Hoechst microplate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50206310(5-Methoxy-9-oxo-9,10-dihydro-acridine-4-carboxylic...)
Affinity DataIC50:  193nMAssay Description:Inhibition of ABCB1 expressed in Kb-V1 cells after 10 mins by calcein-AM assayMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50075373(1N-{4-[2-(6,7-dimethoxy-1,2,3,4-tetrahydro-2-isoqu...)
Affinity DataIC50:  223nMAssay Description:Inhibition of ABCB1 expressed in Kb-V1 cells after 10 mins by calcein-AM assayMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50344754(CHEMBL1779525 | N-{4-[2-(7-Methoxy-6-{2-[2-(2-meth...)
Affinity DataIC50:  390nMAssay Description:Inhibition of ABCG2 expressed in human MCF7/Topo cells by Hoechst microplate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50344752(CHEMBL1777831 | methyl 4-(4-(2-(6-methoxy-7-(2-(2-...)
Affinity DataIC50:  508nMAssay Description:Inhibition of ABCG2 expressed in human MCF7/Topo cells by Hoechst microplate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50075373(1N-{4-[2-(6,7-dimethoxy-1,2,3,4-tetrahydro-2-isoqu...)
Affinity DataIC50:  526nMAssay Description:Inhibition of ABCG2 expressed in human MCF7/Topo cells by Hoechst microplate assayMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50344760(CHEMBL1779519 | N-{4-[2-(6,7-Dimethoxy-3,4-dihydro...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of ABCB1 expressed in Kb-V1 cells after 10 mins by calcein-AM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50344761(CHEMBL1779518 | N-{4-[2-(6,7-Dimethoxy-3,4-dihydro...)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of ABCG2 expressed in human MCF7/Topo cells by Hoechst microplate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50344757(CHEMBL1779522 | N-{4-[2-(6-Methoxy-7-{2-[2-(2-meth...)
Affinity DataIC50: >6.20E+3nMAssay Description:Inhibition of ABCG2 expressed in human MCF7/Topo cells by Hoechst microplate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50293013(CHEMBL455275 | Methyl 4-((4-(2-(6,7-dimethoxy-1,2,...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ABCB1 expressed in Kb-V1 cells after 10 mins by calcein-AM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50293015(CHEMBL502503 | Methyl 4-((4-(2-(6,7-Dimethoxy-1,2,...)
Affinity DataIC50: >2.90E+4nMAssay Description:Inhibition of ABCB1 expressed in Kb-V1 cells after 10 mins by calcein-AM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50344755(CHEMBL1779524 | N-{4-[2-(7-Methoxy-6-{2-[2-(2-meth...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ABCB1 expressed in Kb-V1 cells after 10 mins by calcein-AM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50344761(CHEMBL1779518 | N-{4-[2-(6,7-Dimethoxy-3,4-dihydro...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ABCB1 expressed in Kb-V1 cells after 10 mins by calcein-AM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50344756(CHEMBL1779523 | N-{4-[2-(6-Methoxy-7-{2-[2-(2-meth...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ABCB1 expressed in Kb-V1 cells after 10 mins by calcein-AM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50344758(CHEMBL1779521 | N-{4-[2-(7-Methoxy-6-{2-[2-(2-meth...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ABCB1 expressed in Kb-V1 cells after 10 mins by calcein-AM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50344752(CHEMBL1777831 | methyl 4-(4-(2-(6-methoxy-7-(2-(2-...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ABCB1 expressed in Kb-V1 cells after 10 mins by calcein-AM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50344759(CHEMBL1779520 | N-{4-[2-(7-Methoxy-6-{2-[2-(2-meth...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ABCG2 expressed in human MCF7/Topo cells by Hoechst microplate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50344758(CHEMBL1779521 | N-{4-[2-(7-Methoxy-6-{2-[2-(2-meth...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ABCG2 expressed in human MCF7/Topo cells by Hoechst microplate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50344753(CHEMBL1779526 | N-{4-[2-(6-Methoxy-7-{2-[2-(2-meth...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ABCB1 expressed in Kb-V1 cells after 10 mins by calcein-AM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50344756(CHEMBL1779523 | N-{4-[2-(6-Methoxy-7-{2-[2-(2-meth...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ABCG2 expressed in human MCF7/Topo cells by Hoechst microplate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50344759(CHEMBL1779520 | N-{4-[2-(7-Methoxy-6-{2-[2-(2-meth...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ABCB1 expressed in Kb-V1 cells after 10 mins by calcein-AM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50344757(CHEMBL1779522 | N-{4-[2-(6-Methoxy-7-{2-[2-(2-meth...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ABCB1 expressed in Kb-V1 cells after 10 mins by calcein-AM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50344760(CHEMBL1779519 | N-{4-[2-(6,7-Dimethoxy-3,4-dihydro...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ABCG2 expressed in human MCF7/Topo cells by Hoechst microplate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50344754(CHEMBL1779525 | N-{4-[2-(7-Methoxy-6-{2-[2-(2-meth...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ABCB1 expressed in Kb-V1 cells after 10 mins by calcein-AM assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed