Compile Data Set for Download or QSAR
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Found 13 Enz. Inhib. hit(s) with all data for entry = 50033700
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50349897(CHEMBL1814705)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50349897(CHEMBL1814705)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]U69,593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50349896(CHEMBL1814704)
Affinity DataKi:  67nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50349894(CHEMBL1814702)
Affinity DataKi:  619nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50349895(CHEMBL1814703)
Affinity DataKi:  1.08E+3nMAssay Description:Displacement of [3H]U69,593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50349897(CHEMBL1814705)
Affinity DataKi:  1.23E+3nMAssay Description:Displacement of [3H]DADLE from human recombinant delta opioid receptor expressed in recombinant hDOR-CHO cells after 2 hrs by liquid scintillation co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50349896(CHEMBL1814704)
Affinity DataKi:  1.23E+3nMAssay Description:Displacement of [3H]U69,593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50349896(CHEMBL1814704)
Affinity DataKi:  1.25E+3nMAssay Description:Displacement of [3H]DADLE from human recombinant delta opioid receptor expressed in recombinant hDOR-CHO cells after 2 hrs by liquid scintillation co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50349895(CHEMBL1814703)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]DAMGO from human recombinant mu opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50349895(CHEMBL1814703)
Affinity DataKi: >5.20E+3nMAssay Description:Displacement of [3H]DADLE from human recombinant delta opioid receptor expressed in recombinant hDOR-CHO cells after 2 hrs by liquid scintillation co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50349894(CHEMBL1814702)
Affinity DataKi: >5.20E+3nMAssay Description:Displacement of [3H]DADLE from human recombinant delta opioid receptor expressed in recombinant hDOR-CHO cells after 2 hrs by liquid scintillation co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse And The National Institute On Alcohol Abuse And Alcoholism

Curated by ChEMBL
LigandPNGBDBM50349894(CHEMBL1814702)
Affinity DataKi: >4.00E+4nMAssay Description:Displacement of [3H]U69,593 from human recombinant kappa opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed