Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50033422
TargetSolute carrier family 5 member 4(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM20880((2S,3R,4R,5S,6R)-2-{4-chloro-3-[(4-ethoxyphenyl)me...)
Affinity DataIC50:  1.35nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells using methyl-alpha-D-glucopyranoside by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 5 member 4(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50345019((2R,3S,4R,5R,6S)-2-(hydroxymethyl)-6-(3-(4-(pent-2...)
Affinity DataIC50:  59.5nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells using methyl-alpha-D-glucopyranoside by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 5 member 4(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50345022((2R,3S,4R,5R,6S)-2-Hydroxymethyl-6-(15-oxa-tricycl...)
Affinity DataIC50:  81.9nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells using methyl-alpha-D-glucopyranoside by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 5 member 4(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50345020((2R,3S,4R,5R,6S)-2-Hydroxymethyl-6-(15-oxa-tricycl...)
Affinity DataIC50:  89.6nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells using methyl-alpha-D-glucopyranoside by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 5 member 4(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50345023((2R,3S,4R,5R,6S)-2-Hydroxymethyl-6-(16-oxa-tricycl...)
Affinity DataIC50:  99.7nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells using methyl-alpha-D-glucopyranoside by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 5 member 4(Homo sapiens (Human))
Green Cross

Curated by ChEMBL
LigandPNGBDBM50345021((2R,3S,4R,5R,6S)-2-Hydroxymethyl-6-(16-oxa-tricycl...)
Affinity DataIC50:  103nMAssay Description:Inhibition of human SGLT2 expressed in CHO cells using methyl-alpha-D-glucopyranoside by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed