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Found 31 Enz. Inhib. hit(s) with all data for entry = 50033428
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM20732((4E,6Z,8S,9S,10E,12S,13R,14S,16R)-13-hydroxy-8,14,...)
Affinity DataIC50:  40nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345159(CHEMBL1779539)
Affinity DataIC50:  61nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345167(CHEMBL1779547)
Affinity DataIC50:  78nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50344140(CHEMBL1778208)
Affinity DataIC50:  82nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345150((3aR)-13,13,16-trimethyl-15-oxo-1,2,3,3a,4,5,12,14...)
Affinity DataIC50:  96nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345153(CHEMBL1779533)
Affinity DataIC50:  96nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345155(CHEMBL1779535)
Affinity DataIC50:  106nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50340250((6S)-6,15,15,18-tetramethyl-17-oxo-2,3,4,5,6,7,14,...)
Affinity DataIC50:  110nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345152(CHEMBL1779532)
Affinity DataIC50:  126nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345158(CHEMBL1779538)
Affinity DataIC50:  153nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345165(CHEMBL1779545)
Affinity DataIC50:  170nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345164(CHEMBL1779544)
Affinity DataIC50:  188nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345156(CHEMBL1779536)
Affinity DataIC50:  201nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345163(CHEMBL1779543)
Affinity DataIC50:  301nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345156(CHEMBL1779536)
Affinity DataIC50:  440nMAssay Description:Inhibition of human ERG by HT patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345161(CHEMBL1779541)
Affinity DataIC50:  496nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345160(CHEMBL1779540)
Affinity DataIC50:  634nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345162(CHEMBL1779542)
Affinity DataIC50:  883nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345152(CHEMBL1779532)
Affinity DataIC50:  900nMAssay Description:Inhibition of human ERG by HT patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345166(CHEMBL1779546)
Affinity DataIC50:  982nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345151(CHEMBL1779531)
Affinity DataIC50:  1.04E+3nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345165(CHEMBL1779545)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human ERG by HT patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345150((3aR)-13,13,16-trimethyl-15-oxo-1,2,3,3a,4,5,12,14...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human ERG by HT patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345154(CHEMBL1779534)
Affinity DataIC50:  3.32E+3nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345167(CHEMBL1779547)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of human ERG by HT patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345157(CHEMBL1779537)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of HSP90alpha after 3 hrs by fluorescence polarization binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345153(CHEMBL1779533)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of human ERG by HT patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345159(CHEMBL1779539)
Affinity DataIC50:  1.64E+4nMAssay Description:Inhibition of human ERG by HT patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345150((3aR)-13,13,16-trimethyl-15-oxo-1,2,3,3a,4,5,12,14...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of FYNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345155(CHEMBL1779535)
Affinity DataIC50:  2.44E+4nMAssay Description:Inhibition of human ERG by HT patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50345150((3aR)-13,13,16-trimethyl-15-oxo-1,2,3,3a,4,5,12,14...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of SRC-related membrane-associated tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed