Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 50033526
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50218922(2-Phenyl-2,5-dihydro-pyrazolo[3,4-c]quinolin-4-one...)
Affinity DataKi:  30.8nMAssay Description:Displacement of [125I]I-AB-MECA from human recombinant adenosine A3 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50091117(2-Phenyl-2H-pyrazolo[3,4-c]quinolin-4-ylamine | 2-...)
Affinity DataKi:  91nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50346906(CHEMBL1795497)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50346905(CHEMBL1795495)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50218922(2-Phenyl-2,5-dihydro-pyrazolo[3,4-c]quinolin-4-one...)
Affinity DataKi:  203nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50346907(CHEMBL1795496)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50346908(CHEMBL1795499)
Affinity DataKi:  455nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50346909(CHEMBL1795502)
Affinity DataKi:  500nMAssay Description:Displacement of [125I]I-AB-MECA from human recombinant adenosine A3 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50091117(2-Phenyl-2H-pyrazolo[3,4-c]quinolin-4-ylamine | 2-...)
Affinity DataKi:  551nMAssay Description:Displacement of [125I]I-AB-MECA from human recombinant adenosine A3 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50346910(CHEMBL1795500)
Affinity DataKi:  600nMAssay Description:Displacement of [125I]I-AB-MECA from human recombinant adenosine A3 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50091117(2-Phenyl-2H-pyrazolo[3,4-c]quinolin-4-ylamine | 2-...)
Affinity DataKi:  659nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50346909(CHEMBL1795502)
Affinity DataKi:  750nMAssay Description:Displacement of [3H]ZM241385 from human recombinant adenosine A2A receptor expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50346909(CHEMBL1795502)
Affinity DataKi:  970nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in CHO cell membranes by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed