Compile Data Set for Download or QSAR
maximum 50k data
Found 15 Enz. Inhib. hit(s) with all data for entry = 50033549
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347195(CHEMBL1795747)
Affinity DataIC50:  96nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347200(CHEMBL1795752)
Affinity DataIC50:  190nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50098126(2-(morpholin-4-yl)-benzo[h]chromen-4-one | 2-Morph...)
Affinity DataIC50:  300nMAssay Description:Inhibition of DNA-PKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347198(CHEMBL1795750)
Affinity DataIC50:  330nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50159668(2-Morpholin-4-yl-benzo[g]chromen-4-one | 2-morphol...)
Affinity DataIC50:  400nMAssay Description:Inhibition of DNA-PKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347191(CHEMBL1795743)
Affinity DataIC50:  420nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347194(CHEMBL1795746)
Affinity DataIC50:  717nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347190(CHEMBL1795742)
Affinity DataIC50:  720nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347199(CHEMBL1795751)
Affinity DataIC50:  760nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347197(CHEMBL1795749)
Affinity DataIC50:  930nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347196(CHEMBL1795748)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347193(CHEMBL1795745)
Affinity DataIC50:  2.43E+3nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347201(CHEMBL1795753)
Affinity DataIC50:  3.09E+3nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50159678(3-Morpholin-4-yl-benzo[f]chromen-1-one | 3-morphol...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of DNA-PKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
La Trobe University

Curated by ChEMBL
LigandPNGBDBM50347192(CHEMBL1795744)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of purified DNA-PK by ADP-Glo Kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed