Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 4658
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Riken Advanced Science Institute

LigandPNGBDBM81544(BNS-22)
Affinity DataIC50:  2.80E+3nMpH: 7.5 T: 2°CAssay Description:In vitro inhibition of TOP2 alpha activity by BNS derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Riken Advanced Science Institute

LigandPNGBDBM81549(BNS-65)
Affinity DataIC50:  8.20E+3nMpH: 7.5 T: 2°CAssay Description:In vitro inhibition of TOP2 alpha activity by BNS derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Riken Advanced Science Institute

LigandPNGBDBM81548(BNS-54)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:In vitro inhibition of TOP2 alpha activity by BNS derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Riken Advanced Science Institute

LigandPNGBDBM81547(BNS-53)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:In vitro inhibition of TOP2 alpha activity by BNS derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Riken Advanced Science Institute

LigandPNGBDBM81545(BNS-51)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:In vitro inhibition of TOP2 alpha activity by BNS derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Riken Advanced Science Institute

LigandPNGBDBM81546(BNS-52)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:In vitro inhibition of TOP2 alpha activity by BNS derivatives.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed