Compile Data Set for Download or QSAR
maximum 50k data
Found 34 Enz. Inhib. hit(s) with all data for entry = 50033718
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350161(CHEMBL1814468)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350151(CHEMBL1814458)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50335937(8-Methyl-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-ca...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350152(CHEMBL1814459)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  5.40nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350156(CHEMBL1814463)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350155(CHEMBL1814462)
Affinity DataKi:  8.5nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350160(CHEMBL1814467)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350153(CHEMBL1814460)
Affinity DataKi:  22.9nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350159(CHEMBL1814466)
Affinity DataKi:  29.4nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350161(CHEMBL1814468)
Affinity DataKi:  31.3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350163(CHEMBL1814470)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350158(CHEMBL1814465)
Affinity DataKi:  133nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350152(CHEMBL1814459)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350164(CHEMBL1814471)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350163(CHEMBL1814470)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350160(CHEMBL1814467)
Affinity DataKi:  270nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350154(CHEMBL1814461)
Affinity DataKi:  430nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  790nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350156(CHEMBL1814463)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350157(CHEMBL1814464)
Affinity DataKi:  1.18E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi: >2.82E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350162(CHEMBL1814469)
Affinity DataKi:  3.44E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350164(CHEMBL1814471)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350162(CHEMBL1814469)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350159(CHEMBL1814466)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350151(CHEMBL1814458)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350153(CHEMBL1814460)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50335937(8-Methyl-4-oxo-1-pentyl-1,4-dihydro-quinoline-3-ca...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350154(CHEMBL1814461)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350155(CHEMBL1814462)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350157(CHEMBL1814464)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universita Degli Studi Di Siena

Curated by ChEMBL
LigandPNGBDBM50350158(CHEMBL1814465)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed