Compile Data Set for Download or QSAR
maximum 50k data
Found 13 Enz. Inhib. hit(s) with all data for entry = 50001227
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013923(3-(1-Butyl-4-methoxy-naphthalen-2-yl)-N-(1-methyl-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013924(3-(1-Butyl-4,7-dimethoxy-naphthalen-2-yl)-N-(1-met...)
Affinity DataIC50:  3nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013921(3-(1-Butyl-5-methoxy-naphthalen-2-yl)-N-(1-methyl-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013925(3-(1-Butyl-6-methoxy-naphthalen-2-yl)-N-(1-methyl-...)
Affinity DataIC50:  7nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013922(3-(1-Butyl-7-methoxy-naphthalen-2-yl)-N-(1-methyl-...)
Affinity DataIC50:  15nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013929(3-(6-Methoxy-3-pentyl-benzo[b]thiophen-2-yl)-N-(1-...)
Affinity DataIC50:  24nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013926(CHEMBL319384 | N-(1-Ethyl-4-pyridin-3-yl-butyl)-3-...)
Affinity DataIC50:  26nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013933(3-[6-Methoxy-1-(4-methoxy-phenyl)-3,4-dihydro-naph...)
Affinity DataIC50:  30nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013930(3-(6-Methoxy-3-pentyl-1H-inden-2-yl)-N-(1-methyl-4...)
Affinity DataIC50:  33nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013928(3-(6-Methoxy-3-pentyl-benzofuran-2-yl)-N-(1-methyl...)
Affinity DataIC50:  40nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013927(5-(4-Methoxy-phenyl)-deca-2,4-dienoic acid (1-meth...)
Affinity DataIC50:  40nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013931(3-[6-Methoxy-1-(4-methoxy-phenyl)-naphthalen-2-yl]...)
Affinity DataIC50:  55nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013932(3-(1-Butyl-6-methoxy-3,4-dihydro-naphthalen-2-yl)-...)
Affinity DataIC50:  90nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed