Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 5436
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86341(Phosphodiester analog, 4j | Phosphodiester analog,...)
Affinity DataIC50:  17nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86345(Phosphodiester analog, 6 | Phosphodiester analog, ...)
Affinity DataIC50:  30nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86339(Phosphodiester analog, 4h)
Affinity DataIC50:  55nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86342(Phosphodiester analog, 4k)
Affinity DataIC50:  100nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86340(Phosphodiester analog, 4i)
Affinity DataIC50:  120nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86343(Phosphodiester analog, 4l)
Affinity DataIC50:  130nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86338(Phosphodiester analog, 4g)
Affinity DataIC50:  4.00E+3nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86345(Phosphodiester analog, 6 | Phosphodiester analog, ...)
Affinity DataIC50:  9.00E+3nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86337(Phosphodiester analog, 4f)
Affinity DataIC50:  1.10E+4nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86329(Phosphodiester analog, 3j)
Affinity DataIC50:  1.10E+4nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86341(Phosphodiester analog, 4j | Phosphodiester analog,...)
Affinity DataIC50:  1.20E+4nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86336(Phosphodiester analog, 4e)
Affinity DataIC50:  1.90E+4nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86335(Phosphodiester analog, 4d)
Affinity DataIC50:  3.50E+4nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86318(Phosphodiester analog, 1)
Affinity DataIC50:  3.60E+4nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86344(Phosphodiester analog, 5)
Affinity DataIC50:  4.50E+4nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86327(Phosphodiester analog, 3h)
Affinity DataIC50:  6.60E+4nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86331(Phosphodiester analog, 3l)
Affinity DataIC50:  7.00E+4nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86328(Phosphodiester analog, 3i)
Affinity DataIC50:  9.40E+4nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86330(Phosphodiester analog, 3k)
Affinity DataIC50:  1.54E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86319(Phosphodiester analog, 2)
Affinity DataIC50:  1.74E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86333(Phosphodiester analog, 4b)
Affinity DataIC50: >2.00E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86332(Phosphodiester analog, 4a)
Affinity DataIC50: >2.00E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86326(Phosphodiester analog, 3g)
Affinity DataIC50:  2.00E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86325(Phosphodiester analog, 3f)
Affinity DataIC50: >2.00E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86334(Phosphodiester analog, 4c)
Affinity DataIC50: >2.00E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86323(Phosphodiester analog, 3d)
Affinity DataIC50: >2.00E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86322(Phosphodiester analog, 3c)
Affinity DataIC50: >2.00E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86321(Phosphodiester analog, 3b)
Affinity DataIC50: >2.00E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86320(Phosphodiester analog, 3a)
Affinity DataIC50: >2.00E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
National Cancer Institute-Frederick

LigandPNGBDBM86324(Phosphodiester analog, 3e)
Affinity DataIC50: >2.00E+5nMpH: 8.0 T: 2°CAssay Description:The evaluation of Plk1 PBD binding affinities of the synthetic compounds using an ELISA-based 96-well assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed