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Found 43 Enz. Inhib. hit(s) with all data for entry = 50033750
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136445(5-Chloro-1H-indole-2-carboxylic acid ((R)-2-oxo-1,...)
Affinity DataIC50:  25nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136451(5-Chloro-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50:  25nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136440(5-Bromo-1H-indole-2-carboxylic acid (1-methyl-2-ox...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136437(5-Chloro-1H-indole-2-carboxylic acid (2-oxo-1,2,3,...)
Affinity DataIC50:  44nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136447(5-Chloro-1H-indole-2-carboxylic acid ((S)-2-oxo-1,...)
Affinity DataIC50:  47nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136428(5-Chloro-1H-indole-2-carboxylic acid ((S)-1-methyl...)
Affinity DataIC50:  57nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136448(5-Chloro-1H-indole-2-carboxylic acid ((R)-1-methyl...)
Affinity DataIC50:  61nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136424(5-Chloro-7-fluoro-1H-indole-2-carboxylic acid (1-m...)
Affinity DataIC50:  83nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136450(7-Chloro-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50:  88nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136430(5-Chloro-1H-indole-2-carboxylic acid ((R)-2-oxo-2,...)
Affinity DataIC50:  99nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136416(6-Chloro-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50:  99nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136435(5-Chloro-1H-indole-2-carboxylic acid (2-oxo-2,3,4,...)
Affinity DataIC50:  105nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136425(5-Chloro-1H-indole-2-carboxylic acid (2-oxo-1-pyri...)
Affinity DataIC50:  110nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136443(5-Methyl-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136414(5-Fluoro-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136420(5-Chloro-1H-indole-2-carboxylic acid (2-oxo-1-pyri...)
Affinity DataIC50:  130nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136429(5-Chloro-1H-indole-2-carboxylic acid [1-(5-methyl-...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136418(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-1,2,3,...)
Affinity DataIC50:  160nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136441(5-Chloro-1H-indole-2-carboxylic acid {1-[5-(1H-imi...)
Affinity DataIC50:  160nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136417(5-Cyano-1H-indole-2-carboxylic acid (1-methyl-2-ox...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136442(5-Chloro-1H-indole-2-carboxylic acid ((S)-2-oxo-2,...)
Affinity DataIC50:  240nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136434(7-Nitro-1H-indole-2-carboxylic acid (1-methyl-2-ox...)
Affinity DataIC50:  300nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136444(5-Chloro-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50:  305nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136433(7-Amino-1H-indole-2-carboxylic acid (1-methyl-2-ox...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136419(3,4-Dichloro-N-(2-oxo-1,2,3,4-tetrahydro-quinolin-...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136449(5-Trifluoromethyl-1H-indole-2-carboxylic acid (1-m...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136439(4-Chloro-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136415(5-Methoxy-1H-indole-2-carboxylic acid (1-methyl-2-...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136438(5-Ethyl-1H-indole-2-carboxylic acid (1-methyl-2-ox...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50350687(CHEMBL1814684)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50350688(CHEMBL1814498)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50350692(CHEMBL1814507)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136432(2-(1-Methyl-2-oxo-1,2,3,4-tetrahydro-quinolin-3-yl...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50350694(CHEMBL1504147)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50350693(CHEMBL128249)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136413(3,4-Dichloro-N-(2-oxo-2,3,4,5-tetrahydro-1H-benzo[...)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50350690(CHEMBL128850)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50350691(CHEMBL338902)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50350689(CHEMBL1814500)
Affinity DataIC50:  1.65E+4nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136422(5-Chloro-2-(1-methyl-2-oxo-1,2,3,4-tetrahydro-quin...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136431(5-Phenyl-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136426(6-Phenyl-1H-indole-2-carboxylic acid (1-methyl-2-o...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Applied Science University

Curated by ChEMBL
LigandPNGBDBM50136427(5-Chloro-2-(1-methyl-2-oxo-1,2,3,4-tetrahydro-quin...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human liver glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed