Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 4660
TargetHTH-type transcriptional regulator MgrA(Staphylococcus aureus)
The University Of Chicago

LigandPNGBDBM11979(5-[(3-carboxy-4-hydroxyphenyl)methyl]-2-hydroxyben...)
Affinity DataIC50:  8.00E+3nMpH: 7.4 T: 2°CAssay Description:A fluorescence anisotropy (FA)-based biochemical assay that monitors MgrA-DNA binding. To determine the binding affinity of MgrA to the labeled DNA,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator MgrA(Staphylococcus aureus)
The University Of Chicago

LigandPNGBDBM81554(MgrA inhibitor, 3)
Affinity DataIC50:  2.80E+4nMpH: 7.4 T: 2°CAssay Description:A fluorescence anisotropy (FA)-based biochemical assay that monitors MgrA-DNA binding. To determine the binding affinity of MgrA to the labeled DNA,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator MgrA(Staphylococcus aureus)
The University Of Chicago

LigandPNGBDBM81553(MgrA inhibitor, 2)
Affinity DataIC50:  3.00E+4nMpH: 7.4 T: 2°CAssay Description:A fluorescence anisotropy (FA)-based biochemical assay that monitors MgrA-DNA binding. To determine the binding affinity of MgrA to the labeled DNA,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHTH-type transcriptional regulator MgrA(Staphylococcus aureus)
The University Of Chicago

LigandPNGBDBM81555(MgrA inhibitor, 4)
Affinity DataIC50:  3.20E+4nMpH: 7.4 T: 2°CAssay Description:A fluorescence anisotropy (FA)-based biochemical assay that monitors MgrA-DNA binding. To determine the binding affinity of MgrA to the labeled DNA,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed