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Found 5 Enz. Inhib. hit(s) with all data for entry = 50033798
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50099066(CHEMBL279115 | phorbol 13-acetate 12-myristate)
Affinity DataEC50:  1.70E+6nMAssay Description:Binding affinity to recombinant C1 domain of PKCalpha expressed in Escherichia coli BL21 (DE3) after 45 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50351475(CHEMBL1819528)
Affinity DataEC50:  5.04E+6nMAssay Description:Binding affinity to recombinant C1 domain of PKCalpha expressed in Escherichia coli BL21 (DE3) after 45 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Houston

Curated by ChEMBL
LigandPNGBDBM50351474(CHEMBL1819531)
Affinity DataEC50:  2.98E+6nMAssay Description:Binding affinity to recombinant C1 domain of PKCalpha expressed in Escherichia coli BL21 (DE3) after 45 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Houston

Curated by ChEMBL
LigandPNGBDBM23928(1,3-dimethoxy-5-[(E)-2-(4-methoxyphenyl)ethenyl]be...)
Affinity DataEC50:  1.56E+6nMAssay Description:Binding affinity to recombinant C1 domain of PKCalpha expressed in Escherichia coli BL21 (DE3) after 45 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Houston

Curated by ChEMBL
LigandPNGBDBM23926((E)-resveratrol | 5-[(E)-2-(4-hydroxyphenyl)etheny...)
Affinity DataEC50:  5.78E+6nMAssay Description:Binding affinity to recombinant C1 domain of PKCalpha expressed in Escherichia coli BL21 (DE3) after 45 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed