Compile Data Set for Download or QSAR
maximum 50k data
Found 31 Enz. Inhib. hit(s) with all data for entry = 50034303
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360256(CHEMBL1928201)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360257(CHEMBL1928202)
Affinity DataIC50:  100nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360242(CHEMBL1928218)
Affinity DataIC50:  300nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360241(CHEMBL1928217)
Affinity DataIC50:  450nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360263(CHEMBL1928208)
Affinity DataIC50:  500nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360260(CHEMBL1928205)
Affinity DataIC50:  550nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360249(CHEMBL1928343)
Affinity DataIC50:  660nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360237(CHEMBL1928213)
Affinity DataIC50:  670nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360247(CHEMBL1928341)
Affinity DataIC50:  840nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360267(CHEMBL1928212)
Affinity DataIC50:  960nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360238(CHEMBL1928214)
Affinity DataIC50:  970nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360264(CHEMBL1928209)
Affinity DataIC50:  1.20E+3nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360239(CHEMBL1928215)
Affinity DataIC50:  1.21E+3nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360240(CHEMBL1928216)
Affinity DataIC50:  1.63E+3nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360243(CHEMBL1928219)
Affinity DataIC50:  2.33E+3nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360245(CHEMBL1928339)
Affinity DataIC50:  2.62E+3nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360246(CHEMBL1928340)
Affinity DataIC50:  3.06E+3nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360248(CHEMBL1928342)
Affinity DataIC50:  3.30E+3nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360250(CHEMBL1928344)
Affinity DataIC50:  4.98E+3nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360258(CHEMBL1928203)
Affinity DataIC50:  6.14E+3nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360266(CHEMBL1928211)
Affinity DataIC50:  6.40E+3nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360265(CHEMBL1928210)
Affinity DataIC50:  6.70E+3nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360253(CHEMBL1928347)
Affinity DataIC50:  7.00E+3nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360259(CHEMBL1928204)
Affinity DataIC50:  7.05E+3nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360262(CHEMBL1928207)
Affinity DataIC50:  1.86E+4nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360252(CHEMBL1928346)
Affinity DataIC50:  5.64E+4nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360251(CHEMBL1928345)
Affinity DataIC50:  6.91E+4nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360261(CHEMBL1928206)
Affinity DataIC50:  7.09E+4nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360254(CHEMBL1928348)
Affinity DataIC50:  1.78E+5nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360244(CHEMBL1928338)
Affinity DataIC50:  2.18E+5nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya

Curated by ChEMBL
LigandPNGBDBM50360255(CHEMBL1928349)
Affinity DataIC50:  2.29E+5nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed