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Found 3 Enz. Inhib. hit(s) with all data for entry = 50034191
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
San Diego State University

Curated by ChEMBL
LigandPNGBDBM20732((4E,6Z,8S,9S,10E,12S,13R,14S,16R)-13-hydroxy-8,14,...)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to Hsp90 N-domainMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
San Diego State University

Curated by ChEMBL
LigandPNGBDBM50358580(CHEMBL1923743)
Affinity DataKd:  2.00E+4nMAssay Description:Binding affinity to Hsp90 after 1 hrs by Western blottingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
San Diego State University

Curated by ChEMBL
LigandPNGBDBM50358579(CHEMBL192264)
Affinity DataKd:  1.00E+5nMAssay Description:Binding affinity to human Hsp90 closed state by fluorescence polarization anisotropyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed