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Found 4 Enz. Inhib. hit(s) with all data for entry = 50034517
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363765(CHEMBL1946234)
Affinity DataKi:  144nMAssay Description:Displacement of [3H]mesulergine from human 5HT2C receptor expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363763(CHEMBL342432)
Affinity DataKi:  391nMAssay Description:Displacement of [3H]mesulergine from human 5HT2C receptor expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50035179(Agomelatine | CHEMBL10878 | N-[2-(7-Methoxy-naphth...)
Affinity DataKi:  708nMAssay Description:Displacement of [3H]mesulergine from human 5HT2C receptor expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Lille

Curated by ChEMBL
LigandPNGBDBM50363764(CHEMBL1946233)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]mesulergine from human 5HT2C receptor expressed in CHO cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed