Affinity DataKi: 0.400nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 152nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 153nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 194nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 246nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 391nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 394nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 467nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 474nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 496nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 524nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 575nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 581nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 596nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 682nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 717nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 739nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 910nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 997nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.36E+3nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.82E+3nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.88E+3nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.90E+3nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Arena Pharmaceuticals
Curated by ChEMBL
Arena Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human ERG by patch-clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of CYP1A2 in human liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of CYP2C9 in human liver microsomesMore data for this Ligand-Target Pair