Compile Data Set for Download or QSAR
maximum 50k data
Found 123 Enz. Inhib. hit(s) with all data for entry = 50004613
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataIC50:  3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of wild type Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataIC50:  680nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptase Lys103Asn mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484786(CHEMBL1958457)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50073606(CHEMBL1958265)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of wild type Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50073606(CHEMBL1958265)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50073606(CHEMBL1958265)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50073606(CHEMBL1958265)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptase Lys103Asn mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50073606(CHEMBL1958265)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of ribonuclease H activity of wild type Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484795(CHEMBL1958254)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484827(CHEMBL1958234 | N''-(3,4-Dihydroxybenzylidene)Benz...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50073606(CHEMBL1958265)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of ribonuclease H activity of Human immunodeficiency virus 1 reverse transcriptase Lys103Asn mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484832(CHEMBL1958252)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484824(CHEMBL565153 | NSC-99726)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484824(CHEMBL565153 | NSC-99726)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484795(CHEMBL1958254)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484810(CHEMBL1958255 | NSC-99727)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484813(CHEMBL1958231 | NSC-99722)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM83185(7-[(4-aminobenzoyl)amino]-4-hydroxy-naphthalene-2-...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484785(CHEMBL1958456 | NSC-657715)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM53069(4-[2-(2-pyridinylamino)-4-thiazolyl]benzene-1,2-di...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484833(CHEMBL1958258)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484796(CHEMBL1958256 | NSC-353681)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484808(CHEMBL1958233 | NSC-205497)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484807(CHEMBL1958232 | NSC-204474)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484813(CHEMBL1958231 | NSC-99722)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484839(CHEMBL1958257 | NSC-203867)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484810(CHEMBL1958255 | NSC-99727)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484796(CHEMBL1958256 | NSC-353681)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484785(CHEMBL1958456 | NSC-657715)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484835(CHEMBL1958448)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484797(CHEMBL1955890)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484827(CHEMBL1958234 | N''-(3,4-Dihydroxybenzylidene)Benz...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484833(CHEMBL1958258)
Affinity DataIC50:  5.10E+4nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484788(CHEMBL1958459)
Affinity DataIC50:  5.10E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484811(CHEMBL1958259)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50247434(CHEMBL1958235)
Affinity DataIC50:  5.80E+4nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484777(CHEMBL1958443)
Affinity DataIC50:  5.90E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484809(CHEMBL1958236)
Affinity DataIC50:  6.10E+4nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484812(CHEMBL1958260)
Affinity DataIC50:  6.20E+4nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484797(CHEMBL1955890)
Affinity DataIC50:  6.30E+4nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484834(CHEMBL1958237)
Affinity DataIC50:  6.40E+4nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484802(CHEMBL1958447)
Affinity DataIC50:  6.60E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484812(CHEMBL1958260)
Affinity DataIC50:  6.70E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484839(CHEMBL1958257 | NSC-203867)
Affinity DataIC50:  7.00E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484803(CHEMBL1958451)
Affinity DataIC50:  7.30E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484803(CHEMBL1958451)
Affinity DataIC50:  7.60E+4nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484825(CHEMBL1958263)
Affinity DataIC50:  7.80E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484811(CHEMBL1958259)
Affinity DataIC50:  8.40E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484836(CHEMBL1958458)
Affinity DataIC50:  8.50E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of Human immunodeficiency virus 1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50484798(CHEMBL1958261)
Affinity DataIC50:  9.00E+4nMAssay Description:Inhibition of ribonuclease H activity of HIV1 reverse transcriptase using as poly(dC)-[3H]poly(rG) as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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