Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with all data for entry = 50045932
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM29490(Pyrazolo[1,5-a]-1,3,5-triazine, 13-15)
Affinity DataIC50:  6.10nMAssay Description:Antagonist activity at human CRF1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor-binding protein(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM29490(Pyrazolo[1,5-a]-1,3,5-triazine, 13-15)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity to CRF-binding protein (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed