Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50039714
TargetEstrogen receptor(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50382735(CHEMBL2024377)
Affinity DataIC50:  0.200nMAssay Description:Displacement of [3H]-estradiol from human full length recombinant ERalpha by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50161712((4-Chloro-phenyl)-(4-{4-[6-hydroxy-2-(4-hydroxy-ph...)
Affinity DataIC50:  0.220nMAssay Description:Displacement of [3H]-17beta-estradiol from ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50161706((4-{4-[6-Hydroxy-2-(4-hydroxy-phenyl)-benzo[b]thio...)
Affinity DataIC50:  0.270nMAssay Description:Displacement of [3H]-17beta-estradiol from ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50161698(CHEMBL178334 | [6-Hydroxy-2-(4-hydroxy-phenyl)-ben...)
Affinity DataIC50:  0.280nMAssay Description:Displacement of [3H]-17beta-estradiol from ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50382734(CHEMBL2024376)
Affinity DataIC50:  0.600nMAssay Description:Displacement of [3H]-estradiol from human full length recombinant ERalpha by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50382735(CHEMBL2024377)
Affinity DataIC50:  2.60nMAssay Description:Displacement of [3H]-estradiol from human full length recombinant ERbeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50382734(CHEMBL2024376)
Affinity DataIC50:  3.10nMAssay Description:Displacement of [3H]-estradiol from human full length recombinant ERbeta by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50161712((4-Chloro-phenyl)-(4-{4-[6-hydroxy-2-(4-hydroxy-ph...)
Affinity DataIC50:  9.07nMAssay Description:Displacement of [3H]-17beta-estradiol from ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50161706((4-{4-[6-Hydroxy-2-(4-hydroxy-phenyl)-benzo[b]thio...)
Affinity DataIC50:  12.5nMAssay Description:Displacement of [3H]-17beta-estradiol from ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50161698(CHEMBL178334 | [6-Hydroxy-2-(4-hydroxy-phenyl)-ben...)
Affinity DataIC50:  33.9nMAssay Description:Displacement of [3H]-17beta-estradiol from ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed