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Found 12 Enz. Inhib. hit(s) with all data for entry = 50039567
TargetCytochrome P450 1A1(Rattus norvegicus)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380109(CHEMBL2013099)
Affinity DataIC50:  5.42nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A1(Rattus norvegicus)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380110(CHEMBL2013100)
Affinity DataIC50:  5.53nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A1(Rattus norvegicus)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380107(CHEMBL2013097)
Affinity DataIC50:  5.69nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A1(Rattus norvegicus)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380108(CHEMBL2013098)
Affinity DataIC50:  6.62nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A1(Rattus norvegicus)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380111(CHEMBL2013101)
Affinity DataIC50:  7.74nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A1(Rattus norvegicus)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380106(CHEMBL2013096)
Affinity DataIC50:  8.36nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A1(Rattus norvegicus)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380103(CHEMBL2013093)
Affinity DataIC50:  9.71nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A1(Rattus norvegicus)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380104(CHEMBL2013094)
Affinity DataIC50:  10.4nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A1(Rattus norvegicus)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380105(CHEMBL2013095)
Affinity DataIC50:  13.2nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A1(Rattus norvegicus)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380101(CHEMBL2013091)
Affinity DataIC50:  24.2nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A1(Rattus norvegicus)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380112(CHEMBL2013102)
Affinity DataIC50:  61.4nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A1(Rattus norvegicus)
King Abdulaziz University

Curated by ChEMBL
LigandPNGBDBM50380102(CHEMBL2013092)
Affinity DataIC50:  86.7nMAssay Description:Inhibition of CYP1A1 activity in rat liver microsomes using benzo[alpha]pyrene as substrate after 10 mins by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed