TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant COX2More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of recombinant AKR1C3 assessed as enzyme catalyzed oxidation of S-tetralol by fluorimetric assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Affinity DataIC50: 740nMAssay Description:Inhibition of recombinant COX2More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Affinity DataIC50: 2.23E+3nMAssay Description:Inhibition of recombinant COX1More data for this Ligand-Target Pair
TargetAndrogen receptor(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:Antagonist activity at androgen receptor expressed in HeLa-AR3A-PSA-(ARE)4-Luc13 cells assessed as rightward shift of DHT-induced response incubated ...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C1(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Affinity DataIC50: 6.74E+3nMAssay Description:Inhibition of recombinant AKR1C1 assessed as enzyme catalyzed oxidation of S-tetralol by fluorimetric assayMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C2(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Affinity DataIC50: 8.17E+3nMAssay Description:Inhibition of recombinant AKR1C2 assessed as enzyme catalyzed oxidation of S-tetralol by fluorimetric assayMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C4(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Affinity DataIC50: 8.17E+3nMAssay Description:Inhibition of recombinant AKR1C4 assessed as enzyme catalyzed oxidation of S-tetralol by fluorimetric assayMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C1(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Affinity DataIC50: 1.11E+4nMAssay Description:Inhibition of recombinant AKR1C1 assessed as enzyme catalyzed oxidation of S-tetralol by fluorimetric assayMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C1(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Affinity DataIC50: 2.27E+4nMAssay Description:Inhibition of recombinant AKR1C1 assessed as enzyme catalyzed oxidation of S-tetralol by fluorimetric assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Affinity DataIC50: 3.08E+4nMAssay Description:Inhibition of recombinant COX1More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C4(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Affinity DataIC50: 3.27E+4nMAssay Description:Inhibition of recombinant AKR1C4 assessed as enzyme catalyzed oxidation of S-tetralol by fluorimetric assayMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C4(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Affinity DataIC50: 6.27E+4nMAssay Description:Inhibition of recombinant AKR1C4 assessed as enzyme catalyzed oxidation of S-tetralol by fluorimetric assayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant COX1More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant COX2More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant COX2More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Perelman School Of Medicine University Of Pennsylvania
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant COX1More data for this Ligand-Target Pair