Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 5615
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Frederick National Laboratory For Cancer Research

LigandPNGBDBM91675(Peptide-peptoid hybrid, 6q)
Affinity DataIC50:  15nMAssay Description:Pkk1 PDB fluorescence polarization competition binding assay using Plk. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Frederick National Laboratory For Cancer Research

LigandPNGBDBM91676(Peptide-peptoid hybrid, 7)
Affinity DataIC50:  19nMAssay Description:Pkk1 PDB fluorescence polarization competition binding assay using Plk. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Frederick National Laboratory For Cancer Research

LigandPNGBDBM91677(Peptide-peptoid hybrid, 13)
Affinity DataIC50:  71nMAssay Description:Pkk1 PDB fluorescence polarization competition binding assay using Plk. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed