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Found 18 Enz. Inhib. hit(s) with all data for entry = 50039786
TargetMyeloblastin(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384111(CHEMBL2029556)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384108(CHEMBL2029554)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of cathepsin G using Suc-Ala-Ala-Pro-Phe-p-nitroanilide as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384112(CHEMBL2029557)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human neutrophil elastase using chromogenic substrate (N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384104(CHEMBL2029559)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384111(CHEMBL2029556)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of human neutrophil elastase using chromogenic substrate (N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384108(CHEMBL2029554)
Affinity DataIC50:  1.28E+4nMAssay Description:Inhibition of proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384111(CHEMBL2029556)
Affinity DataIC50:  1.42E+4nMAssay Description:Inhibition of cathepsin G using Suc-Ala-Ala-Pro-Phe-p-nitroanilide as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384112(CHEMBL2029557)
Affinity DataIC50:  1.45E+4nMAssay Description:Inhibition of proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384108(CHEMBL2029554)
Affinity DataIC50:  1.56E+4nMAssay Description:Inhibition of human neutrophil elastase using chromogenic substrate (N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384104(CHEMBL2029559)
Affinity DataIC50:  1.56E+4nMAssay Description:Inhibition of human neutrophil elastase using chromogenic substrate (N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384104(CHEMBL2029559)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of cathepsin G using Suc-Ala-Ala-Pro-Phe-p-nitroanilide as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384112(CHEMBL2029557)
Affinity DataIC50:  3.69E+5nMAssay Description:Inhibition of cathepsin G using Suc-Ala-Ala-Pro-Phe-p-nitroanilide as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384110(CHEMBL2029555)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human neutrophil elastase using chromogenic substrate (N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384109(CHEMBL2029350)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human neutrophil elastase using chromogenic substrate (N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384107(CHEMBL2029553)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human neutrophil elastase using chromogenic substrate (N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384106(CHEMBL2029552)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human neutrophil elastase using chromogenic substrate (N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384105(CHEMBL2029551)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human neutrophil elastase using chromogenic substrate (N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50384113(CHEMBL2029558)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human neutrophil elastase using chromogenic substrate (N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed