Compile Data Set for Download or QSAR
maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 50039973
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387070(CHEMBL2047060)
Affinity DataIC50:  1.62E+3nMAssay Description:Inhibition of human wild type B-Raf kinase assessed as change in ATP consumption by luciferase-luiferin-coupled chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387080(CHEMBL2047071)
Affinity DataIC50:  2.12E+3nMAssay Description:Inhibition of human wild type B-Raf kinase assessed as change in ATP consumption by luciferase-luiferin-coupled chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387081(CHEMBL2047072)
Affinity DataIC50:  2.49E+3nMAssay Description:Inhibition of human wild type B-Raf kinase assessed as change in ATP consumption by luciferase-luiferin-coupled chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387076(CHEMBL2047066)
Affinity DataIC50:  2.74E+3nMAssay Description:Inhibition of human wild type B-Raf kinase assessed as change in ATP consumption by luciferase-luiferin-coupled chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387067(CHEMBL2047057)
Affinity DataIC50:  2.81E+3nMAssay Description:Inhibition of human wild type B-Raf kinase assessed as change in ATP consumption by luciferase-luiferin-coupled chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387079(CHEMBL2047069)
Affinity DataIC50:  3.76E+3nMAssay Description:Inhibition of human wild type B-Raf kinase assessed as change in ATP consumption by luciferase-luiferin-coupled chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387083(CHEMBL2047070)
Affinity DataIC50:  7.48E+3nMAssay Description:Inhibition of human wild type B-Raf kinase assessed as change in ATP consumption by luciferase-luiferin-coupled chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387078(CHEMBL2047068)
Affinity DataIC50:  8.89E+3nMAssay Description:Inhibition of human wild type B-Raf kinase assessed as change in ATP consumption by luciferase-luiferin-coupled chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387075(CHEMBL2047065)
Affinity DataIC50:  9.07E+3nMAssay Description:Inhibition of human wild type B-Raf kinase assessed as change in ATP consumption by luciferase-luiferin-coupled chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387077(CHEMBL2047067)
Affinity DataIC50:  1.35E+4nMAssay Description:Inhibition of human wild type B-Raf kinase assessed as change in ATP consumption by luciferase-luiferin-coupled chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387068(CHEMBL2047058)
Affinity DataIC50:  2.05E+4nMAssay Description:Inhibition of human wild type B-Raf kinase assessed as change in ATP consumption by luciferase-luiferin-coupled chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387069(CHEMBL2047059)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of human wild type B-Raf kinase assessed as change in ATP consumption by luciferase-luiferin-coupled chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387074(CHEMBL2047064)
Affinity DataIC50:  2.27E+4nMAssay Description:Inhibition of human wild type B-Raf kinase assessed as change in ATP consumption by luciferase-luiferin-coupled chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387073(CHEMBL2047063)
Affinity DataIC50:  2.37E+4nMAssay Description:Inhibition of human wild type B-Raf kinase assessed as change in ATP consumption by luciferase-luiferin-coupled chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387066(CHEMBL2047056)
Affinity DataIC50:  2.85E+4nMAssay Description:Inhibition of human wild type B-Raf kinase assessed as change in ATP consumption by luciferase-luiferin-coupled chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387072(CHEMBL2047062)
Affinity DataIC50:  4.51E+4nMAssay Description:Inhibition of human wild type B-Raf kinase assessed as change in ATP consumption by luciferase-luiferin-coupled chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387082(CHEMBL2047073)
Affinity DataIC50:  5.91E+4nMAssay Description:Inhibition of human wild type B-Raf kinase assessed as change in ATP consumption by luciferase-luiferin-coupled chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50387071(CHEMBL2047061)
Affinity DataIC50:  9.16E+4nMAssay Description:Inhibition of human wild type B-Raf kinase assessed as change in ATP consumption by luciferase-luiferin-coupled chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed