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Found 34 Enz. Inhib. hit(s) with all data for entry = 50039975
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  32nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
TargetBeta-secretase 1(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387090(CHEMBL2047229)
Affinity DataIC50:  600nMAssay Description:Inhibition of BACE1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387094(CHEMBL2047224)
Affinity DataIC50:  600nMAssay Description:Inhibition of BACE1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387092(CHEMBL2047227)
Affinity DataIC50:  700nMAssay Description:Inhibition of BACE1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387088(CHEMBL2047375)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of BACE1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387095(CHEMBL2047223)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of BACE1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387092(CHEMBL2047227)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of equine BuChE using butyrylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387095(CHEMBL2047223)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of equine BuChE using butyrylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387091(CHEMBL2047228)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of equine BuChE using butyrylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387094(CHEMBL2047224)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of equine BuChE using butyrylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387093(CHEMBL2047225)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of equine BuChE using butyrylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
TargetBeta-secretase 1(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387093(CHEMBL2047225)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of BACE1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of BACE1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of equine BuChE using butyrylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387088(CHEMBL2047375)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of equine BuChE using butyrylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387097(CHEMBL2047226)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of equine BuChE using butyrylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387090(CHEMBL2047229)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of equine BuChE using butyrylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387089(CHEMBL2047231)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of equine BuChE using butyrylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387095(CHEMBL2047223)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387092(CHEMBL2047227)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387094(CHEMBL2047224)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387093(CHEMBL2047225)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387089(CHEMBL2047231)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of BACE1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387090(CHEMBL2047229)
Affinity DataIC50:  9.40E+3nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387097(CHEMBL2047226)
Affinity DataIC50:  9.90E+3nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387096(CHEMBL2047230)
Affinity DataIC50:  9.90E+3nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387089(CHEMBL2047231)
Affinity DataIC50:  1.03E+4nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387091(CHEMBL2047228)
Affinity DataIC50:  1.11E+4nMAssay Description:Inhibition of BACE1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387096(CHEMBL2047230)
Affinity DataIC50:  1.14E+4nMAssay Description:Inhibition of equine BuChE using butyrylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  1.26E+4nMAssay Description:Inhibition of equine BuChE using butyrylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387088(CHEMBL2047375)
Affinity DataIC50:  1.26E+4nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387091(CHEMBL2047228)
Affinity DataIC50:  1.29E+4nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate after 5 mins by DTNB methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
University Of Waterloo

Curated by ChEMBL
LigandPNGBDBM50387087(CHEMBL2047376)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of BACE1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed