Compile Data Set for Download or QSAR
maximum 50k data
Found 28 Enz. Inhib. hit(s) with all data for entry = 5674
TargetAcetylcholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataKi:  26nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
TargetCholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92554(Coumarin analogue, 3l)
Affinity DataKi:  41nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92543(Coumarin analogue, 3a)
Affinity DataKi:  41nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92545(Coumarin analogue, 3c)
Affinity DataKi:  61nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92544(Coumarin analogue, 3b)
Affinity DataKi:  64nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92548(Coumarin analogue, 3f)
Affinity DataKi:  71nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92553(Coumarin analogue, 3k)
Affinity DataKi:  72nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92551(Coumarin analogue, 3i)
Affinity DataKi:  72nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92549(Coumarin analogue, 3g)
Affinity DataKi:  74nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92550(Coumarin analogue, 3h)
Affinity DataKi:  81nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92546(Coumarin analogue, 3d)
Affinity DataKi:  131nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92547(Coumarin analogue, 3e)
Affinity DataKi:  181nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92552(Coumarin analogue, 3j)
Affinity DataKi:  212nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92548(Coumarin analogue, 3f)
Affinity DataKi:  1.05E+3nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92544(Coumarin analogue, 3b)
Affinity DataKi:  1.25E+3nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92553(Coumarin analogue, 3k)
Affinity DataKi:  1.55E+3nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92547(Coumarin analogue, 3e)
Affinity DataKi:  1.62E+3nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92550(Coumarin analogue, 3h)
Affinity DataKi:  1.81E+3nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92549(Coumarin analogue, 3g)
Affinity DataKi:  2.47E+3nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92546(Coumarin analogue, 3d)
Affinity DataKi:  3.09E+3nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92545(Coumarin analogue, 3c)
Affinity DataKi:  5.41E+3nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92552(Coumarin analogue, 3j)
Affinity DataKi:  5.61E+3nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataKi:  6.32E+3nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92543(Coumarin analogue, 3a)
Affinity DataKi:  7.17E+3nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92554(Coumarin analogue, 3l)
Affinity DataKi:  7.47E+3nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM92551(Coumarin analogue, 3i)
Affinity DataKi:  9.96E+3nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM50022775((m-Hydroxyphenyl)trimethylammonium dimethylcarbama...)
Affinity DataKi:  2.30E+4nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCholinesterase(Homo sapiens (Human))
Comsats Institute Of Information Technology

LigandPNGBDBM50022775((m-Hydroxyphenyl)trimethylammonium dimethylcarbama...)
Affinity DataKi:  4.80E+4nMAssay Description:Inhibition assay using AChE and BuChE.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank