Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 50040513
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM100152(7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)
Affinity DataIC50:  80nMAssay Description:Inhibition of human DYRK1A kinase expressed in Escherichia coli cellsMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM50333423(7-(Pyridin-3-ylmethoxy)-1-methyl-beta-carboline | ...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of DYRK1A kinase using RBER-CHKtide substrate by radiometric protein kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM50395379(CHEMBL2164712 | US9168247, CV12)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DYRK1A kinase using RBER-CHKtide substrate by radiometric protein kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM50333416(7-(2-Methoxyethoxy)-1-methyl-beta-carboline | CHEM...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of DYRK1A kinase using RBER-CHKtide substrate by radiometric protein kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM50395380(CHEMBL2164709 | US9168247, JR84)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of DYRK1A kinase using RBER-CHKtide substrate by radiometric protein kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM50395381(CHEMBL2164716 | US9168247, JR95)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of DYRK1A kinase using RBER-CHKtide substrate by radiometric protein kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
University Of Namur (Fundp)

Curated by ChEMBL
LigandPNGBDBM50395378(CHEMBL2164696 | US9168247, CV24)
Affinity DataIC50:  4.30E+4nMAssay Description:Inhibition of DYRK1A kinase using RBER-CHKtide substrate by radiometric protein kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed