Affinity DataKi: 1.10nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 2.60nMAssay Description:Inverse agonist activity at human recombinant mu opioid receptor expressed in CHO cells after 3 hrs by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20nMAssay Description:Inverse agonist activity at human recombinant mu opioid receptor expressed in CHO cells after 3 hrs by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair