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Found 3 Enz. Inhib. hit(s) with all data for entry = 50040414
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of New England

Curated by ChEMBL
LigandPNGBDBM50297506(CHEMBL551074 | l7-(cyclopropylmethyl)-3,l4-dihydro...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of New England

Curated by ChEMBL
LigandPNGBDBM50297506(CHEMBL551074 | l7-(cyclopropylmethyl)-3,l4-dihydro...)
Affinity DataEC50:  2.60nMAssay Description:Inverse agonist activity at human recombinant mu opioid receptor expressed in CHO cells after 3 hrs by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of New England

Curated by ChEMBL
LigandPNGBDBM50001709(4-cyclopropylmethyl-(13R)-12-oxa-4-azapentacyclo[9...)
Affinity DataEC50:  1.20nMAssay Description:Inverse agonist activity at human recombinant mu opioid receptor expressed in CHO cells after 3 hrs by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed