Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50040129
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50389548(CHEMBL2063990)
Affinity DataIC50:  810nMAssay Description:Inhibition of AKT1 by AKT1/PKBalpha KinEASE FP fluorescein green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50389550(CHEMBL2064009)
Affinity DataIC50:  1.66E+3nMAssay Description:Inhibition of AKT1 by AKT1/PKBalpha KinEASE FP fluorescein green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50389549(CHEMBL2064002)
Affinity DataIC50:  5.02E+3nMAssay Description:Inhibition of AKT1 by AKT1/PKBalpha KinEASE FP fluorescein green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed