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Found 18 Enz. Inhib. hit(s) with all data for entry = 50040233
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhejiang Betapharma

Curated by ChEMBL
LigandPNGBDBM50391089(BPI-2009 | CHEMBL2087361 | Conmana | Icotinib | Lc...)
Affinity DataIC50:  2nMAssay Description:Inhibition of EGFR using GST-Crk as substrate assessed as phosphorylated Crk level after 20 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhejiang Betapharma

Curated by ChEMBL
LigandPNGBDBM50391088(CHEMBL2087360)
Affinity DataIC50:  2nMAssay Description:Inhibition of EGFR using GST-Crk as substrate assessed as phosphorylated Crk level after 20 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhejiang Betapharma

Curated by ChEMBL
LigandPNGBDBM50391086(CHEMBL2087358)
Affinity DataIC50:  2nMAssay Description:Inhibition of EGFR using GST-Crk as substrate assessed as phosphorylated Crk level after 20 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhejiang Betapharma

Curated by ChEMBL
LigandPNGBDBM50391090(CHEMBL2087356)
Affinity DataIC50:  5nMAssay Description:Inhibition of EGFR using GST-Crk as substrate assessed as phosphorylated Crk level after 20 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhejiang Betapharma

Curated by ChEMBL
LigandPNGBDBM50391084(CHEMBL2087355)
Affinity DataIC50:  5nMAssay Description:Inhibition of EGFR using GST-Crk as substrate assessed as phosphorylated Crk level after 20 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhejiang Betapharma

Curated by ChEMBL
LigandPNGBDBM50391085(CHEMBL2087357)
Affinity DataIC50:  7nMAssay Description:Inhibition of EGFR using GST-Crk as substrate assessed as phosphorylated Crk level after 20 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhejiang Betapharma

Curated by ChEMBL
LigandPNGBDBM50391087(CHEMBL2087359)
Affinity DataIC50:  8nMAssay Description:Inhibition of EGFR using GST-Crk as substrate assessed as phosphorylated Crk level after 20 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhejiang Betapharma

Curated by ChEMBL
LigandPNGBDBM50391089(BPI-2009 | CHEMBL2087361 | Conmana | Icotinib | Lc...)
Affinity DataIC50:  45nMAssay Description:Inhibition of EGFR-mediated intracellular tyrosine phosphorylation in EGF-stimulated human A431 cells after 2.5 hrs by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhejiang Betapharma

Curated by ChEMBL
LigandPNGBDBM50391088(CHEMBL2087360)
Affinity DataIC50:  45nMAssay Description:Inhibition of EGFR-mediated intracellular tyrosine phosphorylation in EGF-stimulated human A431 cells after 2.5 hrs by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhejiang Betapharma

Curated by ChEMBL
LigandPNGBDBM50391090(CHEMBL2087356)
Affinity DataIC50:  50nMAssay Description:Inhibition of EGFR-mediated intracellular tyrosine phosphorylation in EGF-stimulated human A431 cells after 2.5 hrs by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhejiang Betapharma

Curated by ChEMBL
LigandPNGBDBM50391084(CHEMBL2087355)
Affinity DataIC50:  50nMAssay Description:Inhibition of EGFR-mediated intracellular tyrosine phosphorylation in EGF-stimulated human A431 cells after 2.5 hrs by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhejiang Betapharma

Curated by ChEMBL
LigandPNGBDBM50391086(CHEMBL2087358)
Affinity DataIC50:  55nMAssay Description:Inhibition of EGFR-mediated intracellular tyrosine phosphorylation in EGF-stimulated human A431 cells after 2.5 hrs by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhejiang Betapharma

Curated by ChEMBL
LigandPNGBDBM50391082(CHEMBL2087353)
Affinity DataIC50:  55nMAssay Description:Inhibition of EGFR using GST-Crk as substrate assessed as phosphorylated Crk level after 20 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhejiang Betapharma

Curated by ChEMBL
LigandPNGBDBM50391080(CHEMBL1198361)
Affinity DataIC50:  85nMAssay Description:Inhibition of EGFR using GST-Crk as substrate assessed as phosphorylated Crk level after 20 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhejiang Betapharma

Curated by ChEMBL
LigandPNGBDBM50391081(CHEMBL2087352)
Affinity DataIC50:  120nMAssay Description:Inhibition of EGFR using GST-Crk as substrate assessed as phosphorylated Crk level after 20 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhejiang Betapharma

Curated by ChEMBL
LigandPNGBDBM50391083(CHEMBL2087354)
Affinity DataIC50:  150nMAssay Description:Inhibition of EGFR using GST-Crk as substrate assessed as phosphorylated Crk level after 20 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhejiang Betapharma

Curated by ChEMBL
LigandPNGBDBM50391087(CHEMBL2087359)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of EGFR-mediated intracellular tyrosine phosphorylation in EGF-stimulated human A431 cells after 2.5 hrs by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Zhejiang Betapharma

Curated by ChEMBL
LigandPNGBDBM50391085(CHEMBL2087357)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of EGFR-mediated intracellular tyrosine phosphorylation in EGF-stimulated human A431 cells after 2.5 hrs by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed