Compile Data Set for Download or QSAR
maximum 50k data
Found 24 Enz. Inhib. hit(s) with all data for entry = 50035857
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50014917(4-(2-Chloro-phenyl)-2-imidazol-1-ylmethyl-6-methyl...)
Affinity DataIC50:  500nMAssay Description:Inhibition of Thromboxane A2 synthase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50368043(CHEMBL1203671)
Affinity DataIC50:  600nMAssay Description:Inhibition of Thromboxane A2 synthase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50014907(4-(2-Difluoromethoxy-phenyl)-2-imidazol-1-ylmethyl...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of Thromboxane A2 synthetase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50368045(CHEMBL1203652)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of Thromboxane A2 synthetase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50368036(CHEMBL1203682)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of Thromboxane A2 synthetase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50368040(CHEMBL1203686)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Thromboxane A2 synthetase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50368033(CHEMBL1203626)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of Thromboxane A2 synthase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50368037(CHEMBL1744226)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of Thromboxane A2 synthase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM7962(4-(2-Imidazol-1-yl-ethoxy)-benzoic acid; hydrochlo...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of Thromboxane A2 synthase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50014918(2-Imidazol-1-ylmethyl-6-methyl-4-(2-nitro-phenyl)-...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of Thromboxane A2 synthetase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50368034(CHEMBL1203674)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of Thromboxane A2 synthetase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50368032(CHEMBL1203662)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of Thromboxane A2 synthase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50368031(CHEMBL1203654)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of Thromboxane A2 synthetase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50368042(CHEMBL1203687)
Affinity DataIC50:  1.18E+4nMAssay Description:Inhibition of Thromboxane A2 synthetase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50368041(CHEMBL1203653)
Affinity DataIC50:  1.28E+4nMAssay Description:Inhibition of Thromboxane A2 synthetase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50014919(4-(2,3-Dichloro-phenyl)-2-imidazol-1-ylmethyl-6-me...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of Thromboxane A2 synthetase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50014908(4-(2-Chloro-3-trifluoromethyl-phenyl)-2-imidazol-1...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of Thromboxane A2 synthetase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50368039(CHEMBL1202293)
Affinity DataIC50:  1.95E+4nMAssay Description:Inhibition of Thromboxane A2 synthase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50368044(CHEMBL1203649)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of Thromboxane A2 synthetase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50014902(4-(2-Difluoromethoxy-phenyl)-2-imidazol-1-ylmethyl...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of Thromboxane A2 synthase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50368038(CHEMBL1203655)
Affinity DataIC50:  7.20E+4nMAssay Description:Inhibition of Thromboxane A2 synthetase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50368035(CHEMBL1203656)
Affinity DataIC50:  1.15E+5nMAssay Description:Inhibition of Thromboxane A2 synthetase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50014915(4-(2-Chloro-3-trifluoromethyl-phenyl)-2-imidazol-1...)
Affinity DataIC50:  1.25E+5nMAssay Description:Inhibition of Thromboxane A2 synthase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50318494(3-ethyl 5-methyl 2,6-dimethyl-4-(3-nitrophenyl)-1,...)
Affinity DataIC50:  1.00E+6nMAssay Description:Inhibition of Thromboxane A2 synthase after oral administration of 0.03 mmol/kgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed