TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
San Francisco State University
Curated by ChEMBL
San Francisco State University
Curated by ChEMBL
Affinity DataIC50: 4.01E+4nMT: 2°CAssay Description:Inhibition of human recombinant SIRT1 using Arg-His-Lys-Lys(epsilon-acetyl)-AMC at room temperature for 45 mins by fluorescent screening assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
San Francisco State University
Curated by ChEMBL
San Francisco State University
Curated by ChEMBL
Affinity DataIC50: 4.58E+4nMAssay Description:Inhibition of human recombinant SIRT2 using Arg-His-Lys-Lys(epsilon-acetyl)-AMC at 37 degC for 45 mins by fluorescent screening assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
San Francisco State University
Curated by ChEMBL
San Francisco State University
Curated by ChEMBL
Affinity DataIC50: 3.70E+6nMT: 2°CAssay Description:Inhibition of human recombinant SIRT1 using Arg-His-Lys-Lys(epsilon-acetyl)-AMC at room temperature for 45 mins by fluorescent screening assayMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
San Francisco State University
Curated by ChEMBL
San Francisco State University
Curated by ChEMBL
Affinity DataIC50: 4.50E+6nMAssay Description:Inhibition of human recombinant SIRT2 using Arg-His-Lys-Lys(epsilon-acetyl)-AMC at 37 degC for 45 mins by fluorescent screening assayMore data for this Ligand-Target Pair