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Found 13 Enz. Inhib. hit(s) with all data for entry = 50004763
TargetElastase(Pseudomonas aeruginosa)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50485657(CHEMBL2146996)
Affinity DataIC50:  2.73E+3nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasB using Abz-Ala-Gly-Leu-Ala-p-Nitro-Benzyl-Amide as substrate incubated for 30 mins prior to substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50485648(CHEMBL2146995)
Affinity DataIC50:  3.34E+3nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasB using Abz-Ala-Gly-Leu-Ala-p-Nitro-Benzyl-Amide as substrate incubated for 30 mins prior to substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50485651(CHEMBL2146997)
Affinity DataIC50:  3.58E+3nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasB using Abz-Ala-Gly-Leu-Ala-p-Nitro-Benzyl-Amide as substrate incubated for 30 mins prior to substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50485646(CHEMBL2146998)
Affinity DataIC50:  4.65E+3nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasB using Abz-Ala-Gly-Leu-Ala-p-Nitro-Benzyl-Amide as substrate incubated for 30 mins prior to substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50485653(CHEMBL2147001)
Affinity DataIC50:  5.27E+3nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasB using Abz-Ala-Gly-Leu-Ala-p-Nitro-Benzyl-Amide as substrate incubated for 30 mins prior to substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50485647(CHEMBL2146999)
Affinity DataIC50:  6.72E+3nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasB using Abz-Ala-Gly-Leu-Ala-p-Nitro-Benzyl-Amide as substrate incubated for 30 mins prior to substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50485654(CHEMBL2147000)
Affinity DataIC50:  8.58E+3nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasB using Abz-Ala-Gly-Leu-Ala-p-Nitro-Benzyl-Amide as substrate incubated for 30 mins prior to substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50015094(CHEMBL152665 | N-Hydroxy-2-phenyl-acetamide | N-hy...)
Affinity DataIC50:  1.36E+4nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasB using Abz-Ala-Gly-Leu-Ala-p-Nitro-Benzyl-Amide as substrate incubated for 30 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50485655(CHEMBL2146994)
Affinity DataIC50:  1.64E+4nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasB using Abz-Ala-Gly-Leu-Ala-p-Nitro-Benzyl-Amide as substrate incubated for 30 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50485649(CHEMBL1650620)
Affinity DataIC50:  8.06E+4nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasB using Abz-Ala-Gly-Leu-Ala-p-Nitro-Benzyl-Amide as substrate incubated for 30 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50485656(CHEMBL1650624)
Affinity DataIC50:  8.85E+4nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasB using Abz-Ala-Gly-Leu-Ala-p-Nitro-Benzyl-Amide as substrate incubated for 30 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50485652(CHEMBL1650621)
Affinity DataIC50:  2.20E+5nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasB using Abz-Ala-Gly-Leu-Ala-p-Nitro-Benzyl-Amide as substrate incubated for 30 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetElastase(Pseudomonas aeruginosa)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50485650(CHEMBL1650623)
Affinity DataIC50:  3.92E+5nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasB using Abz-Ala-Gly-Leu-Ala-p-Nitro-Benzyl-Amide as substrate incubated for 30 mins prior to substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed