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Found 9 Enz. Inhib. hit(s) with all data for entry = 50042496
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50426837(CHEMBL2323142)
Affinity DataIC50:  780nMAssay Description:Inhibition of telomerase-mediated supercoiling activity in human MGC803 cells after 24 hrs by TRAP-PCR-ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50426836(CHEMBL2323143)
Affinity DataIC50:  1.71E+3nMAssay Description:Inhibition of telomerase-mediated supercoiling activity in human MGC803 cells after 24 hrs by TRAP-PCR-ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50426831(CHEMBL2323147)
Affinity DataIC50:  2.11E+3nMAssay Description:Inhibition of telomerase-mediated supercoiling activity in human MGC803 cells after 24 hrs by TRAP-PCR-ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50105463(2,7-diamino-10-ethyl-9-phenylphenanthridinium brom...)
Affinity DataIC50:  2.39E+3nMAssay Description:Inhibition of telomerase-mediated supercoiling activity in human MGC803 cells after 24 hrs by TRAP-PCR-ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50426834(CHEMBL2321890)
Affinity DataIC50:  3.14E+3nMAssay Description:Inhibition of telomerase-mediated supercoiling activity in human MGC803 cells after 24 hrs by TRAP-PCR-ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50426833(CHEMBL2323145)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of telomerase-mediated supercoiling activity in human MGC803 cells after 24 hrs by TRAP-PCR-ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50426835(CHEMBL2323144)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of telomerase-mediated supercoiling activity in human MGC803 cells after 24 hrs by TRAP-PCR-ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50426830(CHEMBL2323141)
Affinity DataIC50:  1.48E+4nMAssay Description:Inhibition of telomerase-mediated supercoiling activity in human MGC803 cells after 24 hrs by TRAP-PCR-ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
Guizhou University

Curated by ChEMBL
LigandPNGBDBM50426832(CHEMBL2323146)
Affinity DataIC50:  2.19E+4nMAssay Description:Inhibition of telomerase-mediated supercoiling activity in human MGC803 cells after 24 hrs by TRAP-PCR-ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed